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Src Family Kinase Inhibitors: Small Molecules and Peptides
24 results for "Src Family Kinase Inhibitors Small Molecules and Peptides" in Products
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Src Family Kinase Inhibitors: Small Molecules and Peptides
24 results for "Src Family Kinase Inhibitors Small Molecules and Peptides" in Products
Catalog #:
6793
Highly potent pan-Src/Bcr-Abl inhibitor
| Alternate Names : | BMS-354825 |
| Chemical Name : | N-(2-Chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-1-piperazinyl]-2-methyl-4-pyrimidinyl]amino]-5-thiazolecarboxamide |
| Purity : | ≥98% (HPLC) |
Inhibits TNF-induced NF-κB activation
| Chemical Name : | 4-[(1E)-2-(3,5-Dihydroxyphenyl)ethenyl]-1,2-benzenediol |
| Purity : | ≥98% (HPLC) |
Catalog #:
5579
Potent and selective breast tumor kinase (Brk) inhibitor
| Chemical Name : | 3-(9H-Pyrido[2,3-b]indol-4-ylamino)phenol |
| Purity : | ≥98% (HPLC) |
Dual Src-Abl inhibitor; antiproliferative
| Alternate Names : | SKI-606 |
| Chemical Name : | 4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methyl-1-piperazinyl)propoxy]-3-quinolinecarbonitrile |
| Purity : | ≥99% |
Potent, selective Src family kinase inhibitor
| Chemical Name : | 1-(1,1-Dimethylethyl)-1-(4-methylphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
| Purity : | ≥99% (HPLC) |
Potent and selective c-Src inhibitor
| Chemical Name : | 1-[3-[1-([1,1'-Biphenyl]-3-ylmethyl)-1H-1,2,3-triazol-5-yl]phenyl]-3-(4-chlorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
| Purity : | ≥98% (HPLC) |
Src family kinase inhibitor; also inhibits c-Abl
| Alternate Names : | 1-NA-PP 1 |
| Chemical Name : | 1-(1,1-Dimethylethyl)-3-(1-naphthalenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
| Purity : | ≥99% (HPLC) |
Potent and selective Lck and Src inhibitor; also inhibits SIK
| Alternate Names : | KIN112 |
| Chemical Name : | 2,6-Dimethylphenyl-N-(2,4-dimethoxyphenyl)-N-[2-[[4-(4-methyl-1-piperazinyl)phenyl]amino]-4-pyrimidinyl]carbamate |
| Purity : | ≥98% (HPLC) |
Src tyrosine kinase inhibitor
| Chemical Name : | N-(2-Chloro-5-methoxyphenyl)-6-methoxy |
| Purity : | ≥99% (HPLC) |
Catalog #:
6981
Selective and highly potent Fgr and Lyn kinase inhibitor; orally bioavailable
| Chemical Name : | 3-[(6,7-Dimethoxy-4-quinazolinyl)oxy]-N-[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-4-methylbenzamide dihydrochloride |
| Purity : | ≥98% (HPLC) |
Catalog #:
6976
Potent PDGFRα and PDGFRβ inhbitor; also inhibits c-Abl, Lck, c-Src and Fyn kinases
| Chemical Name : | N-(3-Fluorophenyl)-1,4-dihydro-6,7-dimethoxyindeno[1,2-c]pyrazol-3-amine |
| Purity : | ≥98% (HPLC) |
Potent c-SRC kinase inhibitor; also inhibits DDR2, BTK and Syk
| Chemical Name : | 3-[[2-[3-(4-Morpholinylmethyl)phenyl]thieno[3,2-b]pyridin-7-yl]amino]phenol dihydrochloride |
| Purity : | ≥98% (HPLC) |
Dual site Src kinase inhibitor
| Chemical Name : | 6,7-Dimethoxy-N-(4-phenoxyphenyl)-4-quinazolinamine |
| Purity : | ≥99% (HPLC) |
Catalog #:
6364
UNC119 chaperone-cargo interaction inhibitor; disrupts Src activation
| Chemical Name : | Ethyl 4-((3,4-dioxo-2-((2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl)amino)cyclobut-1-en-1-yl)amino)piperidine-1-carboxylate hydrochloride |
| Purity : | ≥98% (HPLC) |
Catalog #:
6475
Potent ATP-competitive Src family kinase inhibitor; also AMPK inhibitor; cell permeable
| Chemical Name : | 2,3-Dihydro-N,N-dimethyl-2-oxo-3-[(4,5,6,7-tetrahydro-1H-indol-2-yl)methylene]-1H-indole-5-sulfonamide |
| Purity : | ≥98% (HPLC) |
Inhibitor of Src family kinases
| Chemical Name : | 7-[trans-4-(4-Methyl-1-piperazinyl)cyclohexyl]-5-(4-phenoxyphenyl)-7H-Pyrrolo[2,3-d]pyrimidin-4-amine trihydrochloride |
| Purity : | ≥98% (HPLC) |
Potent, selective Src family kinase inhibitor
| Chemical Name : | 3-(4-chlorophenyl) 1-(1,1-dimethylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
| Purity : | ≥99% (HPLC) |
Catalog #:
3567
Potent Lck inhibitor
| Chemical Name : | 6-(2,6-Dimethylphenyl)-2-[[4-(4-methyl-1-pyrimido[5',4':5,6]pyrimido[1,2-a]benzimidazol-5(6H)-one |
| Purity : | ≥98% (HPLC) |
Potent Src inhibitor; also inhibits FGFR1, PDGFRβ and Wee1
| Chemical Name : | 6-(2,6-Dichlorophenyl)-2-[[4-[2-(diethylamino)ethoxy]phenyl]amino]-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one dihydrochloride |
| Purity : | ≥99% (HPLC) |
Catalog #:
6400
Potent CDK1 and CDK2 inhibitor; also inhibits GSK-3β and Lck
| Chemical Name : | 7,12-Dihydro-9-nitroindolo[3,2-d][1]benzazepin-6(5H)-one |
| Purity : | ≥98% (HPLC) |
Negative control for PP 2 (Cat. No. 1407)
| Chemical Name : | 1-Phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
| Purity : | ≥98% (HPLC) |
Src family kinase inhibitor. Also Hsp90 inhibitor
| Chemical Name : | (15R)-17-demethoxy-15-methoxy-11-O-methyl-geldanamycin |
| Purity : | ≥95% (HPLC) |
Catalog #:
4941
Potent EGFR-kinase inhibitor
| Chemical Name : | 4-[4-[[(1R)-1-Phenylethyl]amino]-7H-pyrrolo[2,3-d]pyrimidin-6-yl]phenol hydrochloride |
| Purity : | ≥98% (HPLC) |
Catalog #:
7189
Potent and selective Src tyrosine kinase family inhibitor; anticancer; antiviral; orally bioavailable
| Alternate Names : | AZD 0530 |
| Chemical Name : | N-(5-Chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methyl-1-piperazinyl)ethoxy]-5-[(tetrahydro-2H-pyran-4-yl)oxy]-4-quinazolinamine |
| Purity : | ≥98% (HPLC) |
