
Methyltransferase Inhibitors Products
23 results for "Methyltransferase Inhibitors" in Products
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Methyltransferase Inhibitors Products
23 results for "Methyltransferase Inhibitors" in Products
Selective PRMT1 inhibitor
Chemical Name : | N,N'-(Sulfonyldi-4,1-phenylene)bis(2-chloroacetamide) |
Purity : | ≥98% (HPLC) |
DNA methyltransferase inhibitor
Chemical Name : | 4-Amino-1-β-D-ribofuranosyl-1,3,5-triazin-2(1H)-one |
Purity : | ≥98% (HPLC) |
Potent and selective PRMT 4 inhibitor
Chemical Name : | N-Methyl-N-((2-(1-(2-(methylamino)ethyl)piperidin-4-yl)pyridin-4-yl)methyl)-3-phenoxybenzamide |
Purity : | ≥98% (HPLC) |
Potent and selective PRMT5 inhibitor
Alternate Names : | EPZ015866, GSK 3203591 |
Chemical Name : | 2-(Cyclobutylamino)-N-[(2S)-3-(3,4-dihydro-2(1H)-isoquinolinyl)-2-hydropropyl]-4-pyridinecarboxamide dihydrochloride |
Purity : | ≥97% (HPLC) |
DNA methyltransferase and cytidine deaminase inhibitor
Alternate Names : | NSC 309132 |
Chemical Name : | 1-β-D-Ribofuranosyl-2(1H)-pyrimidinone |
Purity : | ≥99% (HPLC) |
Allosteric inhibitor of PRMT3
Chemical Name : | N-1,2,3-Benzothiadiazol-6-yl-N'-[2-oxo-2-(1-piperidinyl)ethyl]urea |
Purity : | ≥99% (HPLC) |
DNA methyltransferase inhibitor
Alternate Names : | 2'-Deoxy-5-azacytidine, 5-Aza-2'-deoxycytidine, NSC 127716 |
Chemical Name : | 4-Amino-1-(2-deoxy-β-D-erythro-pentofuranosyl)-1,3,5-triazin-2(1H)-one |
Purity : | ≥99% (HPLC) |
Non-nucleoside DNA methyltransferase inhibitor
Chemical Name : | N-Phthalyl-L-tryptophan |
Purity : | ≥99% (HPLC) |
Potent and selective SETD7 inhibitor
Chemical Name : | 8-Fluoro-1,2,3,4-tetrahydro-N-[(1R)-2-oxo-2-(1-pyrrolidinyl)-1-[[3-(trifluoromethyl)phenyl]methyl]ethyl]-6-isoquinolinesulfonamide hydrochloride |
Purity : | ≥97% (HPLC) |
High affinity and selective WDR5 antagonist
Chemical Name : | N-[2-(4-Methylpiperazin-1-yl)-5-[3-(morpholin-4-ylmethyl)phenyl]phenyl]-6-oxo-4-(trifluoromethyl)-1,6-dihydropyridine-3-carboxamide |
Purity : | ≥98% (HPLC) |
MGMT inhibitor
Alternate Names : | PaTrin-2 |
Chemical Name : | 6-[(4-Bromo-2-thienyl)methoxy]-9H-purin-2-amine |
Purity : | ≥98% (HPLC) |
Potent and selective allosteric inhibitor of PRMT3
Chemical Name : | 1-(Isoquinolin-6-yl)-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl] urea |
Purity : | ≥98% (HPLC) |
Potent and selective PRMT5 inhibitor
Chemical Name : | N-[(2S)-3-(3,4-Dihydro-2(1H)-isoquinolinyl)-2-hydroxypropyl]-6-(3-oxetanylamino)-4-pyrimidinecarboxamide |
Purity : | ≥98% (HPLC) |
WDR5 antagonist
Chemical Name : | 3-[(3-Methoxybenzoyl)amino]-4-(4-methyl-1-piperazinyl)benzoic acid methyl ester |
Purity : | ≥99% (HPLC) |
Negative control of SGC 707 (Cat. No. 5367)
Chemical Name : | N-2-Naphthalenyl-N'-[2-oxo-2-(1-pyrrolidinyl)ethyl]urea |
Purity : | ≥98% (HPLC) |
Selective PRMT1 inhibitor
Chemical Name : | 4,4'-(2,5-Furandiyl)bis-benzenecarboximidamide dihydrochloride |
Purity : | ≥98% (HPLC) |
Highly potent DOT1L inhibitor
Chemical Name : | 7-[5-Deoxy-5-[[3-[[[[4-(1,1-dimethylethyl)phenyl]amino]carbonyl]amino]propyl](1-methylethyl)amino]-β-D-ribofuranosyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
Purity : | ≥98% (HPLC) |
Potent WDR5/MLL interaction inhibitor
Chemical Name : | 1-[[(2S)-5-[(Aminoiminomethyl)amino]-2-[[2-ethyl-2-[(2-methyl-1-oxopropyl)amino]-1-oxobutyl]amino]-1-oxopentyl]amino]-N-[bis(4-fluorophenyl)methyl]-cyclopentanecarboxamide trifluoroacetate |
Purity : | ≥98% (HPLC) |
Potent and selective type I PRMT inhibitor
Chemical Name : | N1-Methyl-N1-[[4-[4-(1-methylethoxy)phenyl]-1H-pyrrol-3-yl]methyl]-1,2-ethanediamine dihydrochloride |
Purity : | ≥98% (HPLC) |
SUV39H1 inhibitor
Chemical Name : | (3S,3'S,5aR,5aR,10bR,10'bR,11aS,11'aS)-2,2',3,3',5a,5'a,6,6'-octahydro-3,3'-bis(hydroxymethyl)-2,2'-dimethyl-[10b,10'b(11H,11'H)-bi3,11a-epidithio-11aH-pyrazino[1',2':1,5]pyrrolo[2,3-b]indole]-1,1',4,4'-tetrone |
Purity : | ≥95% (HPLC) |
Negative control of (R)-PFI 2 hydrochloride (Cat. No. 4892)
Chemical Name : | 8-Fluoro-1,2,3,4-tetrahydro-N-[(1S)-2-oxo-2-(1-pyrrolidinyl)-1-[[3-(trifluoromethyl)phenyl]methyl]ethyl]-6-isoquinolinesulfonamide hydrochloride |
Purity : | ≥97% (HPLC) |
Highly potent and selective DOT1L inhibitor; cell permeable
Chemical Name : | 1-[3-[[[(2R,3S,4R,5R)-5-(4-Amino-5-bromo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-3,4-dihydroxytetrahydrofuran-2-yl]methyl](isopropyl)amino]propyl]-3-[4-(2,2-dimethylethyl)phenyl]urea |
Purity : | ≥99% (HPLC) |