22 results for "P2X Receptor Antagonists Small Molecules and Peptides" in Products
P2X Receptor Antagonists: Small Molecules and Peptides
Potent and selective P2X antagonist
| Chemical Name: | 2',3'-O-(2,4,6-Trinitrophenyl)adenosine-5'-triphosphate tetra(triethylammonium) salt |
| Purity: | ≥95% (HPLC) |
Non-selective P2 antagonist
| Chemical Name: | Pyridoxalphosphate-6-azophenyl-2',4'-disulfonic acid tetrasodium salt |
Potent and selective P2X7 antagonist
| Chemical Name: | N-[1-[[(Cyanoamino)(5-quinolinylamino)methylene]amino]-2,2-dimethylpropyl]-3,4-dimethoxybenzeneacetamide |
| Purity: | ≥97% (HPLC) |
Non-selective P2X antagonist
| Chemical Name: | Pyridoxalphosphate-6-azophenyl-2',5'-disulfonic acid tetrasodium salt |
Potent and selective P2X4 antagonist
| Chemical Name: | 5-(3-Bromophenyl)-1,3-dihydro-2H-benzofuro[3,2-e]-1,4-diazepin-2-one |
| Purity: | ≥98% (HPLC) |
Competitive P2X7 antagonist
| Chemical Name: | 3-[[5-(2,3-Dichlorophenyl)-1H-tetrazol-1-yl]methyl]pyridine hydrochloride |
| Purity: | ≥98% (HPLC) |
Potent and selective P2X7 antagonist; brain penetrant
| Chemical Name: | 2-(Phenylthio)-N-[[tetrahydro-4-(4-phenyl-1-piperazinyl)-2H-pyran-4-yl]methyl-3-pyridinecarboxamide |
| Purity: | ≥98% (HPLC) |
Potent and selective P2X1 antagonist
| Chemical Name: | 8,8'-[Carbonylbis(imino-4,1-phenylenecarbonylimino-4,1-phenylenecarbonylimino)]bis-1,3,5-naphthalenetrisulfonic acid hexasodium salt |
| Purity: | ≥95% (HPLC) |
Potent P2X7 antagonist
| Chemical Name: | N-[2-[[2-[(2-Hydroxyethyl)amino]ethyl]amino]-5-quinolinyl]-2-tricyclo[3.3.1.13,7]dec-1-ylacetamide dihydrochloride |
| Purity: | ≥98% (HPLC) |
Selective and competitive P2X1 antagonist
| Chemical Name: | 8,8'-[carbonylbis(imino-3,1-phenylenecarbonylimino)]bis-1,3,5-naphthalene-trisulphonic acid, hexasodium salt |
Selective P2Y11 and P2X1 antagonist
| Chemical Name: | 8,8'-[Carbonylbis[imino-3,1-phenylenecarbonylimino(4-fluoro-3,1-phenylene)carbonylimino]]bis-1,3,5-naphthalenetrisulfonic acid hexasodium salt |
| Purity: | ≥90% (HPLC) |
Non-competitive P2X7 antagonist
| Chemical Name: | 4-[(2S)-2-[(5-isoquinolinylsulfonyl)methylamino]-3-oxo-3-(4-phenyl-1-piperazinyl)propyl] phenyl isoquinolinesulfonic acid ester |
| Purity: | ≥98% (HPLC) |
Potent and selective P2X7 antagonist
| Chemical Name: | N-Cyano-N"-[(1S)-1-phenylethyl]-N'-5-quinolinyl-guanidine |
| Purity: | ≥98% (HPLC) |
Selective, high affinity P2X3 and P2X2/3 antagonist; antinociceptive
| Chemical Name: | 5-[[[(3-Phenoxyphenyl)methyl][(1S)-1,2,3,4-tetrahydro-1-naphthalenyl]amino]carbonyl]-1,2,4-benzenetricarboxylic acid disodium salt |
| Purity: | ≥98% (HPLC) |
Selective P2X4 antagonist
| Chemical Name: | N-[3-(Aminosulfonyl)-4-(3-chlorophenoxy)phenyl]benzeneacetamide |
| Purity: | ≥98% (HPLC) |
Non-selective P2 antagonist
| Chemical Name: | 8,8'-[Carbonylbis[imino-3,1-phenylenecarbonylimino(4-methyl-3,1-phenylene)carbonylimino]]bis-1,3,5-naphthalenetrisulfonic acid hexasodium salt |
| Purity: | ≥98% (HPLC) |
Dye for assessing cell viability and blood brain barrier permeability; also EAAT inhibitor and iGluR antagonist
| Chemical Name: | 6,6-[(3,3'-Dimethyl[1,1'-biphenyl]-4,4'-diyl)bis(azo)bis[4-amino- 5-hydroxy-1,3-naphthalenedisulphonic acid] tetrasodium salt |
| Purity: | ≥90% (HPLC) |
Potent and selective human P2X7 antagonist
| Chemical Name: | 3-[1-[[(3'-Nitro[1,1'-biphenyl]-4-yl)oxy]methyl]-3-(4-pyridinyl)propyl]-2,4-thiazolidinedione |
| Purity: | ≥98% (HPLC) |
Selective P2X4 allosteric antagonist
| Chemical Name: | N-[2,6-Dibromo-4-(1-methylethyl)phenyl]-N'-(3-pyridinyl)urea |
| Purity: | ≥98% (HPLC) |
Selective P2X3 and P2X2/3 antagonist
| Chemical Name: | 5-[[4,5-Dimethoxy-2-(methylethyl)phenyl]methyl]-2,4-pyrimidinediamine |
| Purity: | ≥98% (HPLC) |
Potent P2X3 antagonist
| Chemical Name: | 4,4',4'',4'''-[Carbonylbis[imino-5,1,3-benzenetriylbis(carbonylimino)]]tetrakisbenzenesulfonic acid tetrasodium salt |
| Purity: | ≥90% (HPLC) |
Highly selective P2X1 antagonist
| Chemical Name: | 4,4',4'',4'''-[Carbonylbis(imino-5,1,3-benzenetriyl-bis(carbonylimino))]tetrakis-1,3-benzenedisulfonic acid, octasodium salt |
| Purity: | ≥90% (HPLC) |
