Methyltransferase Inhibitors Small Molecules and Peptides

WDR5 antagonist

DNA methyltransferase inhibitor

SUV39H1 inhibitor

Non-nucleoside DNA methyltransferase inhibitor

Potent and selective SETD7 inhibitor

Selective PRMT1 inhibitor

Potent and selective PRMT 4 inhibitor

Non-nucleoside DNA methyltransferase inhibitor

MGMT inhibitor

High affinity and selective WDR5 antagonist

High affinity and selective WDR5 antagonist

Potent and selective allosteric inhibitor of PRMT3

Negative control of (R)-PFI 2 hydrochloride (Cat. No. 4892)

Negative control of SGC 707 (Cat. No. 5367)

Highly potent DOT1L inhibitor

Highly potent and selective DOT1L inhibitor; cell permeable

Potent and selective type I PRMT inhibitor

Potent and selective PRMT5 inhibitor

Selective ASH1L histone methyltransferase inhibitor

Selective ASH1L histone methyltransferase inhibitor

Selective ASH1L histone methyltransferase inhibitor