
Other Transferase Inhibitors: Small Molecules and Peptides
23 results for "Other Transferase Inhibitors Small Molecules and Peptides" in Products
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Other Transferase Inhibitors: Small Molecules and Peptides
23 results for "Other Transferase Inhibitors Small Molecules and Peptides" in Products
Thymidylate synthetase inhibitor, also inhibits dihydrofolate reductase, GARFT and AICART
Chemical Name : | N-[4-[2-(2-Amino-4,7-dihydro-4-oxo-3H-pyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoyl]-L-glutamic acid |
Purity : | ≥98% (HPLC) |
Antibiotic; GlcNAc phosphotransferase inhibitor
Chemical Name : | Tunicamycin from Streptomyces sp. |
Purity : | ≥98% (HPLC) |
Inhibitor of γ-glutamyl transpeptidase (GGT)
Chemical Name : | 3-[[(3-Amino-3-carboxypropyl)methoxyphosphinyl]oxy]benzeneacetic acid |
Purity : | ≥95% (HPLC) |
Carnitine palmitoyltransferase I (CPT1) inhibitor
Chemical Name : | (R)-(+)-2-[6-(4-Chlorophenoxy)hexyl]-oxirane-2-carboxylic acid sodium salt |
Purity : | ≥98% (HPLC) |
Potent glutaminyl cyclase inhibitor; disrupts binding of SIRP-α to CD47
Chemical Name : | 6'-Fluoro-2-[4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-piperidinyl]-3,3'-bipyridine |
Purity : | ≥98% (HPLC) |
Nicotinamide N-methyltransferase (NNMT) inhibitor; promotes myoblast differentiation
Chemical Name : | 5-Amino-1-methylquinolinium iodide |
Purity : | ≥97% (HPLC) |
Sialic acid analog; sialyltransferase inhibitor
Chemical Name : | 5-(acetylamino)-3,5-dideoxy-3-fluoro-D-erythro-α-L-manno-2-nonulopyranosonic acid methyl ester 2,4,7,8,9-pentaacetate |
Purity : | ≥97% (HPLC) |
O-GlcNAc transferase (OGT) inhibitor
Chemical Name : | 2-[(4-Chlorophenyl)imino]tetrahydro-4-oxo-3-(2-tricyclo[3.3.1.13,7]dec-1-ylethyl)-2H-1,3-thiazine-6-carboxylic acid |
Purity : | ≥98% (HPLC) |
Potent NLRP3 inflammasome inhibitor; inhibits IL-1β production
Alternate Names : | CP-456773, MCC 950 |
Chemical Name : | N-[[(1,2,3,5,6,7-Hexahydro-s-indacen-4-yl)amino]carbonyl]-4-(1-hydroxy-1-methylethyl)-2-furansulfonamide sodium salt |
Purity : | ≥98% (HPLC) |
α-glucosidase I and II inhibitor; also inhibits ceramide-specific glycosyltransferases and exhibits broad spectrum antiviral activity
Alternate Names : | N-Butyldeoxynojirimycin hydrochloride, NB-DNJ |
Chemical Name : | (2R,3R,4R,5S)-1-Butyl-2-(hydroxymethyl)-3,4,5-piperidinetriol hydrochloride |
Selective p300/CBP inhibitor
Chemical Name : | 4-[4-[[5-(4,5-Dimethyl-2-nitrophenyl)-2-furanyl]methylene]-4,5-dihydro-3-methyl-5-oxo-1H-pyrazol-1-yl]benzoic acid |
Purity : | ≥98% (HPLC) |
Potent FBPase inhibitor; promotes HSC expansion
Chemical Name : | P-[5-[2-Amino-5-(2-methylpropyl)-4-thiazolyl]-2-furanyl]phosphonic acid |
Purity : | ≥98% (HPLC) |
Potent SHMT inhibitor
Chemical Name : | 6-Amino-1,4-dihydro-4-[5-(hydroxymethyl)[1,1'-biphenyl]-3-yl]-3-methyl-4-(1-methylethyl)pyrano[2,3-c]pyrazole-5-carbonitrile |
Purity : | ≥98% (HPLC) |
Potent and selective monoacyglycerol acyltransferase 2 (MOGAT2) inhibitor
Chemical Name : | 7-[4,6-Bis(1,1-dimethylethyl)-2-pyrimidinyl]-5,6,7,8-tetrahydro-3-[4-(trifluoromethoxy)phenyl]-1,2,4-triazolo[4,3-a]pyrazine |
Purity : | ≥98% (HPLC) |
N-acetyltransferase 10 (NAT10) inhibitor
Chemical Name : | 4-[2-(2-Cyclopentylidenehydrazinyl)-4-thiazolyl]benzonitrile |
Purity : | ≥99% (HPLC) |
Potent serine palmitoyltransferase inhibitor
Chemical Name : | rel-1-[1-[2-[(3aR,6aS)-Hexahydrocyclopenta[c]pyrrol-2(1H)-yl]-2-oxoethyl]-4-piperidinyl]-2,3-dihydro-N-methyl-2-oxo-1H-indole-5-carboxamide |
Purity : | ≥98% (HPLC) |
Potent serine palmitoyl transferase inhibitor
Chemical Name : | 4-[6-(1-Oxoheptyl)imidazo[1,2-a]pyridin-8-yl]benzeneacetic acid |
Purity : | ≥98% |
GABA-T inhibitor
Alternate Names : | (±)-γ-Vinyl GABA |
Chemical Name : | 4-Aminohexenoic acid |
Purity : | ≥98% (HPLC) |
Carnitine palmitoyltransferase 1 and 2 (CPT1/2) inhibitor
Chemical Name : | 2-(2,2-Dicyclohexylethyl)piperidine maleate |
Purity : | ≥99% (HPLC) |
Geranylgeranyltransferase I (GGTase I) inhibitor
Chemical Name : | N-[4-[2(R)-Amino-3-mercaptopropyl]amino-2-(1-naphthalenyl)benzoyl]-L-leucine methyl ester trifluoroacetate salt |
Purity : | ≥95% (HPLC) |
Oligosaccharyltransferase (OST) inhibitor; anti-flaviviral
Chemical Name : | 5-[(Dimethylamino)sulfonyl]-N-(5-methyl-2-thiazolyl)-2-(1-pyrrolidinyl)benzamide |
Purity : | ≥98% (HPLC) |
Inhibitor of sphingosine N-acyltransferase
Chemical Name : | 1,1'-[(1S,2R)-1-[(2S,4R,9R,11S,12S)-12-Amino-4,9,11-trihydroxy-2-methyltridecyl]-2-[(1R)-1-methylpentyl]-1,2-ethanediyl-1,2,3-(2R,2'R)-propanetricarboxylic acid ester. |
ICMT inhibitor; arrests cell-cycle at G1 phase
Chemical Name : | 5-(3-Methylphenyl)-1-octyl-1H-indole-3-acetamide |
Purity : | ≥98% (HPLC) |