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EGF Receptor Inhibitors: Small Molecules and Peptides
31 results for "EGF Receptor Inhibitors Small Molecules and Peptides" in Products
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EGF Receptor Inhibitors: Small Molecules and Peptides
31 results for "EGF Receptor Inhibitors Small Molecules and Peptides" in Products
Catalog #:
7371
Potent HER2 receptor tyrosine kinase and EGFR kinase inhibitor
| Chemical Name : | (2E)-N-[4-[[3-Chloro-4-(2-pyridinylmethoxy)phenyl]amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide |
| Purity : | ≥98% (HPLC) |
Catalog #:
7194
Potent, reversible EGFR tyrosine kinase inhibitor
| Chemical Name : | N-(3-Ethynylphenyl)-6,7-bis(2-methoxyethoxy)-4-quinazolinamine hydrochloride |
| Purity : | ≥98% (HPLC) |
Orally active, selective EGFR inhibitor
| Alternate Names : | Gefitinib, ZD 1839 |
| Chemical Name : | N-(3-Chloro-4-fluorophenyl)-7-methoxy-6-[3-(4-morpholinyl)propoxy]-4-quinazolinamine |
| Purity : | ≥98% (HPLC) |
Potent dual specificity EGFR/HER2 inhibitor; active in vivo
| Alternate Names : | BIBW2992 |
| Chemical Name : | (2E)-N-[4-[(3-Chloro-4-fluorophenyl)amino]-7-[[(3S)-tetrahydro-3-furanyl]oxy]-6-quinazolinyl]-4-(dimethylamino)-2-butenamide dimaleate |
| Purity : | ≥98% (HPLC) |
Potent ErbB receptor family inhibitor
| Chemical Name : | N4-(3-Bromophenyl)-N6-methyl-pyrido[3,4-d]pyrimidine-4,6-diamine |
| Purity : | ≥99% (HPLC) |
Catalog #:
6811
Potent and selective dual ErbB2 (HER-2) and EGFR inhibitor
| Chemical Name : | N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine |
| Purity : | ≥98% (HPLC) |
Catalog #:
7640
Potent and selective ErbB2 inhibitor
| Chemical Name : | N6-(4,5-Dihydro-4,4-dimethyl-2-oxazolyl)-N4-[3-methyl-4-([1,2,4]triazolo[1,5-a]pyridin-7-yloxy)phenyl]-4,6-quinazolinediamine |
| Purity : | ≥98% (HPLC) |
Catalog #:
7497
Potent VEGFR-2 inhibitor, also inhibits EGFR and RET oncoproteins activity
| Chemical Name : | N-(4-Bromo-2-fluorophenyl)-6-methoxy-7-[(1-methyl-4-piperidinyl)methoxy]-4-quinazolinamine |
| Purity : | ≥98% (HPLC) |
Catalog #:
6290
Potent mutant-selective EGFR inhibitor
| Chemical Name : | N-[3-[[5-Chloro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-4-pyrimidinyl]oxy]phenyl]-2-propenamide |
| Purity : | ≥98% (HPLC) |
Catalog #:
TB3000-RMU
Iressa synthesized to Ancillary Material Grade
| Chemical Name : | N-(3-Chloro-4-fluorophenyl)-7-methoxy-6-[3-(4-morpholinyl)propoxy]-4-quinazolinamine |
| Purity : | ≥98% |
EGFR kinase inhibitor. Also estrogen and PPARγ ligand
| Chemical Name : | 5,7-Dihydroxy-3-(4-hydroxyphenyl)-4H-1-benzopyran-4-one |
| Purity : | ≥98% (HPLC) |
Potent EGFR and VEGFR inhibitor
| Chemical Name : | 6-[4-[(4-Ethyl-1-piperazinyl)methyl]phenyl]-N-[(1R)-1-phenylethyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
| Purity : | ≥98% (HPLC) |
Catalog #:
6231
Potent irreversible pan ErbB inhibitor
| Alternate Names : | PF00299804 |
| Chemical Name : | (2E)-N-[4-[(3-Chloro-4-fluorophenyl)amino]-7-methoxy-6-quinazolinyl]-4-(1-piperidinyl)-2-butenamide |
| Purity : | ≥98% (HPLC) |
Catalog #:
3580
Dual irreversible inhibitor of ErbB2 and EGFR
| Chemical Name : | (2E)-N-[[4-[[(3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide |
| Purity : | ≥98% (HPLC) |
Catalog #:
3352
Potent ErbB receptor family inhibitor
| Chemical Name : | 5E-4-Amino-6-(4-benzyloxy-3-chlorophenylamino)pyrimidine-5-carboxaldehyde N-(2-morpholin-4-ylethyl) oxime hydrochloride |
| Purity : | ≥97% (HPLC) |
Catalog #:
3599
Potent and selective ErbB2 inhibitor
| Alternate Names : | Mubritinib |
| Chemical Name : | 1-[4-[4-[[2-[(1E)-2-[4-(trifluoromethyl)phenyl]ethenyl]-4-oxazolyl]methoxy]phenyl]butyl]-1H-1,2,3-triazole |
| Purity : | ≥99% (HPLC) |
Highly potent EGFR-kinase inhibitor
| Alternate Names : | Tyrphostin AG 1478 |
| Chemical Name : | N-(3-Chlorophenyl)-6,7-dimethoxy-4-quinazolinanine hydrochloride |
| Purity : | ≥98% (HPLC) |
Potent dual EGFR/ErbB2 inhibitor; orally active
| Chemical Name : | N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[2-[[[2-(methylsulfonyl)ethyl]amino]methyl]-4-thiazolyl]-4-quinazolinamine dihydrochloride |
| Purity : | ≥97% (HPLC) |
EGFR-kinase inhibitor
| Alternate Names : | ZM 252868 |
| Chemical Name : | 4-[(3-Bromophenyl)amino]-6,7-dimethoxyquinazoline hydrochloride |
Selective ErbB2 inhibitor
| Alternate Names : | Tyrphostin AG 825 |
| Chemical Name : | 3-[3-[(2-Benzothiazolylthio)methyl]-4-hydroxy-5-methoxyphenyl]-2-cyano-2-propenamide |
EGFR-kinase inhibitor. Also JAK2, JAK3 inhibitor
| Alternate Names : | Tyrphostin AG 490 |
| Chemical Name : | (E)-2-Cyano-3-(3,4-dihydrophenyl)-N-(phenylmethyl)-2-propenamide |
| Purity : | ≥99% (HPLC) |
Catalog #:
0618
Potent EGFR-kinase inhibitor
| Alternate Names : | Tyrphostin AG 555 |
| Chemical Name : | (E)-2-Cyano-3-(3,4-dihydroxyphenyl)-N-(3-phenylpropyl)-2-propenamide |
| Purity : | ≥99% (HPLC) |
Catalog #:
6349
Potent and irreversible EGFR inhibitor; orally bioavailable
| Alternate Names : | EKB-569 |
| Chemical Name : | (2E)-N-[4-[(3-Chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide |
| Purity : | ≥97% (HPLC) |
Catalog #:
3115
JAK3 kinase inhibitor. Also inhibits EGFR
| Chemical Name : | 2-Bromo-4-[(6,7-dimethoxy-4-quinazolinyl)amino]phenol |
| Purity : | ≥99% (HPLC) |
Highly selective EGFR-kinase inhibitor
| Chemical Name : | N8-(3-Chloro-4-fluorophenyl)-N2-(1-methyl-4-piperidinyl)-pyrimido[5,4-d]pyrimidine-2,8-diamine dihydrochloride |
| Purity : | ≥97% (HPLC) |
