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MEK Inhibitors: Small Molecules and Peptides
11 results for "MEK Inhibitors Small Molecules and Peptides" in Products
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MEK Inhibitors: Small Molecules and Peptides
11 results for "MEK Inhibitors Small Molecules and Peptides" in Products
Potent, selective inhibitor of MEK1 and 2
| Chemical Name : | 1,4-Diamino-2,3-dicyano-1,4-bis[2-aminophenylthio]butadiene |
Potent inhibitor of MEK1/2
| Alternate Names : | PD325901 |
| Chemical Name : | N-[(2R)-2,3-Dihydroxypropoxy]-3,4-difluoro-2-[(2-fluoro-4-iodophenyl)amino]-benzamide |
| Purity : | ≥99% (HPLC) |
Potent MEK1 inhibitor. Also inhibits IκBα phosphorylation
| Alternate Names : | (-)-Arctigenin |
| Chemical Name : | (3R,4R)-4-[(3,4-Dimethoxyphenyl)methyl]dihydro-3-[(4-hydroxy-3-methoxyphenyl)methyl]-2(3H)-furanone |
| Purity : | ≥98% (HPLC) |
Selective MEK inhibitor
| Alternate Names : | CI-1040 |
| Chemical Name : | 2-[(2-Chloro-4-iodophenyl)amino]-N-cyclopropylmethoxy)-3,4-difluorobenzamide |
Catalog #:
7709
Potent and selective MEK inhibitor; orally bioavailable
| Chemical Name : | N-[3-[3-Cyclopropyl-5-[(2-fluoro-4-iodophenyl)amino]-3,4,6,7-tetrahydro-6,8-dimethyl-2,4,7-trioxopyrido[4,3-d]pyrimidin-1(2H)-yl]phenyl]acetamide |
| Purity : | ≥98% (HPLC) |
Selective inhibitor of MEK1 and MEK2; brain penetrant
| Chemical Name : | α-[Amino[(4-aminophenyl)thio]methylene]-2-(trifluoromethyl)benzeneacetonitrile |
| Purity : | ≥99% (HPLC) |
Catalog #:
4824
MEK1 inhibitor
| Chemical Name : | N-[5-[3,4-Difluoro-2-[(2-fluoro-4-iodophenyl)amino]phenyl]-1,3,4-oxadiazol-2-yl]-4-morpholineethanamine |
| Purity : | ≥98% (HPLC) |
Selective MEK5 and ERK5 inhibitor
| Chemical Name : | (3Z)-3-[[[3-[(Dimethylamino)methyl]phenyl]amino]phenylmethylene]-2,3-dihydro-N,N-dimethyl-2-oxo-1H-indole-6-carboxamide |
| Purity : | ≥98% (HPLC) |
MEK inhibitor
| Chemical Name : | 2-(2-Amino-3-methoxyphenyl)-4H-1-benzopyran-4-one |
| Purity : | ≥98% (HPLC) |
Selective inhibitor of MEK1/2
| Chemical Name : | N-(Cyclopropylmethoxy)-3,4,5-trifluoro-2-[(4-iodo-2-methylphenyl)amino]-benzamide |
| Purity : | ≥98% (HPLC) |
Inactive analog of U0126 (Cat. No. 1144)
| Chemical Name : | Bis[amino(methylthio)methylene]butanedinitrile |
