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Histamine H1 Receptor Antagonists: Small Molecules and Peptides

Histamine H1R (HRH1) is a G-protein coupled 7-transmembrane putative glycoprotein that is implicated in the pathogenesis of asthma and is a major pharmaceutical target for antihistamines. It has been detected as a mixture of monomers and homodimers, with highest concentration in the placenta, followed by brain, lung (produced by airway smooth muscle, bronchial epithelium and macrophages) and other tissues.

11 results for "Histamine H1 Receptor Antagonists Small Molecules and Peptides" in Products

Histamine H1 Receptor Antagonists: Small Molecules and Peptides

Histamine H1R (HRH1) is a G-protein coupled 7-transmembrane putative glycoprotein that is implicated in the pathogenesis of asthma and is a major pharmaceutical target for antihistamines. It has been detected as a mixture of monomers and homodimers, with highest concentration in the placenta, followed by brain, lung (produced by airway smooth muscle, bronchial epithelium and macrophages) and other tissues.

11 results for "Histamine H1 Receptor Antagonists Small Molecules and Peptides" in Products

H1 antagonist

Orally active, potent H1 antagonist; also KV11.1 (hERG) channel blocker

H1 antagonist. Also KV11.1 (hERG) and Kir6 (KATP) channel blocker

Selective M2 antagonist

Potent 5-HT2 antagonist; also 5-HT3, H1 and α2 antagonist; antidepressant

Peripheral H1 antagonist; antiallergic agent

H1 receptor antagonist; non-sedating antiallergic agent

H1 antagonist; ocular antiallergic agent

Human pregnane X receptor agonist; H1 antagonist

H1 antagonist

H1 antagonist

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