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Histamine H1 Receptor Antagonists Products
Histamine H1R (HRH1) is a G-protein coupled 7-transmembrane putative glycoprotein that is implicated in the pathogenesis of asthma and is a major pharmaceutical target for antihistamines. It has been detected as a mixture of monomers and homodimers, with highest concentration in the placenta, followed by brain, lung (produced by airway smooth muscle, bronchial epithelium and macrophages) and other tissues.
11 results for "Histamine H1 Receptor Antagonists" in Products
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Histamine H1 Receptor Antagonists Products
Histamine H1R (HRH1) is a G-protein coupled 7-transmembrane putative glycoprotein that is implicated in the pathogenesis of asthma and is a major pharmaceutical target for antihistamines. It has been detected as a mixture of monomers and homodimers, with highest concentration in the placenta, followed by brain, lung (produced by airway smooth muscle, bronchial epithelium and macrophages) and other tissues.
11 results for "Histamine H1 Receptor Antagonists" in Products
H1 antagonist
| Chemical Name : | (2R)-2-[2-[(1R)-1-(4-Chlorophenylethoxy]ethyl]-1-methyl-2-pyrrolidine fumarate |
| Purity : | ≥98% (HPLC) |
Orally active, potent H1 antagonist; also KV11.1 (hERG) channel blocker
| Alternate Names : | Hismanal |
| Chemical Name : | 1-[(4-Fluorophenyl)methyl]-N-[1-[2-(4-methoxyphenyl)ethyl]-4-piperidinyl]-1H-benzimidazol-2-amine |
| Purity : | ≥99% (HPLC) |
H1 antagonist. Also KV11.1 (hERG) and Kir6 (KATP) channel blocker
| Chemical Name : | α-[4-(1,1-Dimethylethyl)phenyl]-4-(hydroxydiphenylmethyl)-1-piperidinebutanol |
| Purity : | ≥98% (HPLC) |
Selective M2 antagonist
| Chemical Name : | N,N-Dimethyl-3-[(1S)-1-(2-pyridinyl)ethyl]-1H-indene-2-ethanamine maleate |
| Purity : | ≥99% (HPLC) |
Potent 5-HT2 antagonist; also 5-HT3, H1 and α2 antagonist; antidepressant
| Alternate Names : | Org 3770, 6-Azamianserin |
| Chemical Name : | 1,2,3,4,10,14b-Hexahydro-2-methylpyrazino[2,1-a]pyrido[2,3-c][2]benzazepine |
| Purity : | ≥99% (HPLC) |
Catalog #:
1944
Peripheral H1 antagonist; antiallergic agent
| Alternate Names : | SCH 29851 |
| Chemical Name : | 4-(8-Chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)-1-piperidinecarboxylic acid ethyl ester |
| Purity : | ≥99% (HPLC) |
H1 receptor antagonist; non-sedating antiallergic agent
| Alternate Names : | MDL 16455, Terfenidine |
| Chemical Name : | α,α-Dimethyl-4-[1-hydroxy-4-[4-(hydroxydiphenylmethyl)-1-piperidinyl]butyl]-benzeneacetic acid hydrochloride |
| Purity : | ≥99% (HPLC) |
Catalog #:
4241
H1 antagonist; ocular antiallergic agent
| Chemical Name : | (Z)-11-[3-(Dimethylamino)propylidene]-6,11-dihydro-dibenz[b,e]oxepin-2-acetic acid hydrochloride |
| Purity : | ≥99% (HPLC) |
Human pregnane X receptor agonist; H1 antagonist
| Alternate Names : | Meclozine |
| Chemical Name : | 1-[(4-Chlorophenyl)phenylmethyl]4-[(3-methylphenyl)methyl]piperazine dihydrochloride |
| Purity : | ≥99% (HPLC) |
Catalog #:
0784
H1 antagonist
| Chemical Name : | 4,9-Dihydro-4-(1-methyl-4-piperidinylidene-10H-benzo[4,5]cyclohepta[1,2-b]thiophen-10-one fumarate |
| Purity : | ≥99% (HPLC) |
Catalog #:
3072
H1 antagonist
| Alternate Names : | DPH |
| Chemical Name : | 2-Diphenylmethoxy-N,N-dimethylethanamine hydrochloride |
| Purity : | ≥99% (HPLC) |
