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23 results for "GABA-A R alpha 1" in Products

GABA-A R alpha 1 Products

GABA A (γ-aminobutyric acid-type A) receptors are members of the cysteine-loop family of neurotransmitter-gated ion channels. GABA binding to A-type receptors induces anion-selective ion channel opening. These receptors are the principal fast inhibitory neurotransmitter receptors in the CNS. GABA A receptors are heteropentamer combinations of seven subunit types; α, β, γ, δ, ε, θ, and π. Three subunits, α, β, and γ, have at least ...

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Competitive and selective GABAA antagonist

Alternate Names:
Gabazine
Chemical Name:
6-Imino-3-(4-methoxyphenyl)-1(6H)-pyridazinebutanoic acid hydrobromide
Purity:
≥98%
Competitive and selective GABAA antagonist
Reactivity:
Human, Mouse, Rat
Details:
Rabbit IgG Polyclonal
Applications:
KO, IHC, WB, ICC/IF, IP
Western Blot: GABA-AR alpha 1 Antibody [NB300-191]

Potent GABAA agonist; also GABAA-ρ partial agonist

Chemical Name:
5-Aminomethyl-3-hydroxyisoxazole
Purity:
≥98%
Potent GABAA agonist; also GABAA-ρ partial agonist

Benzodiazepine partial inverse agonist

Chemical Name:
8-Azido-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylic acid ethyl ester
Purity:
≥98%
Benzodiazepine partial inverse agonist

CNS stimulant

Alternate Names:
PTZ
Chemical Name:
6,7,8,9-Tetrahydro-5H-tetrazolo[1,5-a]azepine
Purity:
≥98%
CNS stimulant
Reactivity:
Mouse, Rat
Details:
Rabbit IgG Polyclonal
Applications:
KO, IHC, WB, IP
Western Blot: GABA-AR alpha 1 Antibody [NB300-207]

Benzodiazepine inverse agonist

Chemical Name:
N-Methyl-β-carboline-3-carboxamide
Purity:
≥99%
Benzodiazepine inverse agonist

GABAA agonist

Alternate Names:
Gaboxadol
Chemical Name:
4,5,6,7-Tetrahydroisoxazolo[5,4-c]pyridin-3-ol hydrochloride
Purity:
≥98%
GABAA agonist

Positive allosteric modulator of GABAA receptors

Alternate Names:
3a,5a-THPROG
Chemical Name:
(3α,5α)-3-Hydroxy-pregnan-20-one
Positive allosteric modulator of GABAA receptors
Reactivity:
Human, Rat
Details:
Rabbit IgG Polyclonal
Applications:
IHC, WB
Western Blot: GABA-AR alpha 1 Antibody [NBP2-16565]
(3)

Benzodiazepine antagonist

Alternate Names:
Ro 15-1788
Chemical Name:
8-Fluoro-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylic acid, ethyl ester
Purity:
≥99%
Benzodiazepine antagonist
Reactivity:
Human
R&D Systems VersaClone cDNA Plasmids

Benzodiazepine inverse agonist

Chemical Name:
4-Ethyl-6,7-dimethoxy-9H-pyrido[3,4-b]indole-3-carboxylic acid methyl ester hydrochloride
Purity:
≥98%
Benzodiazepine inverse agonist

GABAA partial agonist; displays subtype selectivity

Chemical Name:
3-(2,5-Difluorophenyl)-7-(1,1-dimethylethyl)-6-[(1-methyl-1H-1,2,4-triazol-5-yl)methoxy]-1,2,4-triazolo[4,3-b]pyridazine
Purity:
≥98%
GABAA partial agonist; displays subtype selectivity

Postitive allosteric modulator of GABAA receptors

Chemical Name:
(3α,5β)-3-Hydroxy-pregnan-20-one
Postitive allosteric modulator of GABAA receptors

α5-selective GABAA inverse agonist

Chemical Name:
6,7-Dihydro-3-[(2-hydroxyethyl)thio]-6,6-dimethyl-1-(2-thiazolyl)-benzo[c]thiophen-4(5H)-one
Purity:
≥98%
α5-selective GABAA inverse agonist

Active metabolite of oxcarbazepine (Cat. No. 3864)

Alternate Names:
GP 47779
Chemical Name:
10,11-Dihydro-10-hydroxy-5H-dibenz(Z)[b,f]azepin-5-carboxamide
Purity:
≥98%
Active metabolite of oxcarbazepine (Cat. No. 3864)
Reactivity:
Human
Details:
Rabbit IgG Polyclonal
Applications:
WB
Western Blot: GABA-AR alpha 1 Antibody [NBP2-33762]
Reactivity:
Human
Applications:
WB
Western Blot: GABA-AR alpha 1 Overexpression Lysate [NBL1-10915]

Recombinant Monoclonal Antibody

Reactivity:
Human
Details:
Rabbit IgG Kappa Monoclonal Clone #1F4
Applications:
ICC/IF, WB
GABA-AR alpha 1 Antibody (1F4) - Chimeric - Azide and BSA Free

Recombinant Monoclonal Antibody

Reactivity:
Human
Details:
Mouse IgG2b Kappa Monoclonal Clone #1F4
Applications:
ICC/IF, WB
Novus Antibodies
Reactivity:
Human
Source:
E. coli
Applications:
AC
Reactivity:
Human
Details:
Mouse IgG2a Kappa Monoclonal Clone #D4
Applications:
ELISA
Novus Antibodies
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