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Protein Kinase A Inhibitors Products

The cAMP-dependent protein kinase (PKA) holoenzyme is composed of two regulatory and two catalytic subunits, designated PKA R and PKA C, respectively. Upon PKA R subunit binding to the second messenger cAMP, active PKA C subunits are released, initiating a phosphorylation cascade that regulates such cellular functions as metabolism, ion transport, and gene transcription. Catalytic PKA subunit isoforms, Cα, Cβ and, in humans, Cγ, have been identified.

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8 results for "Protein Kinase A Inhibitors" in Products

8 results for "Protein Kinase A Inhibitors" in Products

Protein Kinase A Inhibitors Products

The cAMP-dependent protein kinase (PKA) holoenzyme is composed of two regulatory and two catalytic subunits, designated PKA R and PKA C, respectively. Upon PKA R subunit binding to the second messenger cAMP, active PKA C subunits are released, initiating a phosphorylation cascade that regulates such cellular functions as metabolism, ion transport, and gene transcription. Catalytic PKA subunit isoforms, Cα, Cβ and, in humans, Cγ, have been identified.

View small molecule Protein Kinase A Inhibitors, peptide Protein Kinase A Inhibitors and citations by using the filter on the left, or choose one of the products below to view details.

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Cell-permeable protein kinase A inhibitor

Alternate Names: Protein kinase inhibitor-(14-22)-amide,myristoylated
Purity: ≥95% (HPLC)
Cell-permeable protein kinase A inhibitor

Protein kinase A inhibitor

Chemical Name: N-[2-[[3-(4-Bromophenyl)-2-propenyl]amino]ethyl]-5-isoquinolinesulfonamide dihydrochloride
Purity: ≥98% (HPLC)
Protein kinase A inhibitor

High affinity PKA inhibitor

Purity: ≥95% (HPLC)
High affinity PKA inhibitor

Selective protein kinase A inhibitor

Chemical Name: (9R,10S,12S)-2,3,9,10,11,12-Hexahydro-10-hydroxy-9-methyl-1-oxo-9,12-epoxy-1H-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-10-carboxylic acid, hexyl ester
Purity: ≥97% (HPLC)
Selective protein kinase A inhibitor

Inhibitor of cyclic nucleotide dependent- and Rho-kinases

Alternate Names: HA 1077
Purity: ≥98% (HPLC)
Inhibitor of cyclic nucleotide dependent- and Rho-kinases

Potent pan-Akt and PKA inhibitor

Chemical Name: 4-(4-Chlorophenyl)-4-[4-(1H-pyrazol-4-yl)phenyl]piperidine hydrochloride
Purity: ≥98% (HPLC)
Potent pan-Akt and PKA inhibitor

cAMP antagonist

Chemical Name: (R)-Adenosine, cyclic 3',5'-(hydrogenphosphorothioate) triethylammonium
Purity: ≥98% (HPLC)
cAMP antagonist

Staurosporine synthesized to Ancillary Material Grade

Chemical Name: [9S-(9α,10β,11β,13α)]-2,3,10,11,12,13-Hexahydro-10-methoxy-9-methyl-11-(methylamino)-9,13-epoxy-1H,9H-diindolo[1,2,3-gh:3',2',1'-lm]pyrrolo[3,4-j][1,7]benzodiazonin-1-one
Purity: ≥98%
Staurosporine synthesized to Ancillary Material Grade
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