
Insulin and Insulin-like Receptor Inhibitors: Small Molecules and Peptides
8 results for "Insulin and Insulin-like Receptor Inhibitors Small Molecules and Peptides" in Products
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Insulin and Insulin-like Receptor Inhibitors: Small Molecules and Peptides
8 results for "Insulin and Insulin-like Receptor Inhibitors Small Molecules and Peptides" in Products
Potent and selective dual inhibitor of the IGF-1 receptor and insulin receptor
Chemical Name : | cis-3-[8-Amino-1-(2-phenyl-7-quinolinyl)imidazo[1,5-a]pyrazin-3-yl]-1-methylcyclobutanol |
Purity : | ≥98% (HPLC) |
Potent IR and IGF1R inhibitor; also inhibits anaplastic lymphoma kinase (ALK)
Chemical Name : | 2-[[2-[[1-[(Dimethylamino)ethanoyl]-5-(methyloxy)-2,3-dihydro-1H-indol-6-yl]amino]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino]-6-fluoro-N-methylbenzamide |
Purity : | ≥98% (HPLC) |
High affinity insulin-like growth factor-I binding protein IGFBP inhibitor
Chemical Name : | 1-(3,4-Dihydroxybenzoyl)-6,7-dihydroxy-3-isoquinolinecarboxylic acid |
Purity : | ≥98% (HPLC) |
ATP-competitive inhibitor of IGF1R
Chemical Name : | 5-[3-(Phenylmethoxy)phenyl]-7-[trans-3-(1-pyrrolidinylmethyl)cyclobutyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
Purity : | ≥99% (HPLC) |
IGF1R inhibitor
Chemical Name : | N-(5-Chloro-2-methoxyphenyl)-N'-(2-methyl-4-quinolinyl)urea |
Purity : | ≥99% (HPLC) |
Highly potent ALK inhibitor; also potently inhibits IR, IGF1R, STK22D and FLT3
Alternate Names : | LDK378 |
Chemical Name : | 5-Chloro-N4-[2-[(1-methylethyl)sulfonyl]phenyl]-N2-[5-methyl-2-(1-methylethoxy)-4-(4-piperidinyl)phenyl]-2,4-pyrimidinediamine |
Purity : | ≥98% (HPLC) |
Dual IR/IGF1R inhibitor
Chemical Name : | 4-[[(2S)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino]-3-[7-methyl-5-(4-morpholinyl)-1H-benzimidazol-2-yl]-2(1H)-pyridinone |
Purity : | ≥98% (HPLC) |
Selective IGF1R inhibitor
Alternate Names : | Picropodophyllin |
Chemical Name : | (5R,5aS,8aR,9R)-5,8,8a,9-Tetrahydro-9-hydroxy-5-(3,4,5-trimethoxyphenyl)-furo[3',4':6,7]naphtho[2,3-d]-1,3-dioxol-6(5aH)-one |
Purity : | ≥97% (HPLC) |