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GluR1 Products

GluR1 is a 4-transmembrane protein that belongs to the glutamate-gated ion channel family. It is one of four AMPA receptor subunits that form a functional heterotetrameric glutamate receptor. GluR1 only interacts with GluR2. In addition to constitutive phosphorylation on a key serine in the C-terminal extracellular region, neurotransmitter-induced phosphorylation of another key serine by CaMKII leads to a potentiation of glutamate-mediated current.

14 results for "GluR1" in Products

GluR1 Products

GluR1 is a 4-transmembrane protein that belongs to the glutamate-gated ion channel family. It is one of four AMPA receptor subunits that form a functional heterotetrameric glutamate receptor. GluR1 only interacts with GluR2. In addition to constitutive phosphorylation on a key serine in the C-terminal extracellular region, neurotransmitter-induced phosphorylation of another key serine by CaMKII leads to a potentiation of glutamate-mediated current.

14 results for "GluR1" in Products

Catalog #: RDC1110

Positive allosteric modulator of AMPA receptors; inhibits AMPA desensitization

Broad spectrum glutamatergic antagonist

Potent AMPA antagonist; more selective than CNQX (Cat. No. 0190)

AMPA agonist; also group I mGlu agonist

Selective non-competitive AMPA antagonist

GluK1 antagonist; inhibits carbonic anhydrase (CA) II and IV; also positive allosteric modulator of GABAA receptors

Selective positive allosteric modulator of AMPA receptors

Open-channel blocker of AMPA currents; selective for non-GluA2-containing receptors

Competitive non-NMDA iGluR antagonist

Positive allosteric modulator of AMPA receptors

Non-competitive non-NMDA iGluR antagonist

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