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16 results for "casein-kinase-2-inhibitors&view=expanded" in Products

High affinity, selective CK2 inhibitor

Chemical Name:
3-[[5-(4-Methylphenyl)thieno[2,3-d]pyrimidin-4-yl]thio]propanoic acid
Purity:
≥98%
High affinity, selective CK2 inhibitor

Selective inhibitor of p38 MAPK

Alternate Names:
Adezmapimod
Chemical Name:
4-[5-(4-Fluorophenyl)-2-[4-(methylsulfonyl)phenyl]-1H-imidazol-4-yl]pyridine
Purity:
≥98%
Selective inhibitor of p38 MAPK

Potent p38 MAPK inhibitor; anti-inflammatory

Chemical Name:
N-[4-[2-Ethyl-4-(3-methylphenyl)-5-thiazolyl]-2-pyridinyl]benzamide
Purity:
≥98%
Potent p38 MAPK inhibitor; anti-inflammatory

CK1 inhibitor

Chemical Name:
N-(2-Aminoethyl)-5-chloro-8-isoquinolinesulfonamide dihydrochloride
Purity:
≥99%
CK1 inhibitor

Cdk inhibitor; potently inhibits cdk1 and cdk2; also inhibits CK1; acts as molecular glue

Chemical Name:
(2R)-2-[[9-(Methylethyl)-6-[[[4-(2-pyridinyl)phenyl]methyl]amino]-9H-purin-2-yl]amino]-1-butanol trihydrochloride
Purity:
≥98%
Cdk inhibitor; potently inhibits cdk1 and cdk2; also inhibits CK1; acts as molecular glue

Potent CK1 inhibitor; also inhibits cyclin-dependent kinases

Chemical Name:
2-[[9-(1-Methylethyl)-6-[[3-(2-pyridinyl)phenyl]amino]-9H-purin-2-yl]amino]-1-butanol dihydrochloride
Purity:
≥98%
Potent CK1 inhibitor; also inhibits cyclin-dependent kinases

Selective CK1 inhibitor. Also inhibits TGF-βRI

Chemical Name:
4-[4-(2,3-Dihydro-1,4-benzodioxin-6-yl)-5-(2-pyridinyl)-1H-imidazol-2-yl]benzamide
Purity:
≥98%
Selective CK1 inhibitor. Also inhibits TGF-βRI

Selective cell-permeable CK2 inhibitor

Alternate Names:
NSC 231634
Chemical Name:
4,5,6,7-Tetrabromobenzotriazole
Purity:
≥98%
Selective cell-permeable CK2 inhibitor

Potent and selective CK1ε and CK1δ inhibitor

Chemical Name:
4-[1-Cyclohexyl-4-(4-fluorophenyl)-1H-imidazol-5-yl]-2-pyrimidinamine dihydrochloride
Purity:
≥98%
Potent and selective CK1ε and CK1δ inhibitor

Potent and selective CK1α, CK1δ and CK1ε inhibitor

Chemical Name:
4-(1-((4-Fluoro-1-methylpiperidin-4-yl)methyl)-4-(5-fluoropyridin-2-yl)-1H-imidazol-5-yl)-1H-pyrrolo[2,3-b]pyridine
Purity:
≥98%
Potent and selective CK1α, CK1δ and CK1ε inhibitor
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