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9 results for "Casein Kinase 1 Inhibitors Small Molecules and Peptides" in Products

Casein Kinase 1 Inhibitors: Small Molecules and Peptides

Casein kinase I (CK1) is a monomeric serine-threonine protein kinase with 7 isoforms: α, β, γ1, γ2, γ3, δ and ε. CK1 is involved in a number of cellular processes including DNA repair, cell division, nuclear localization and membrane transport.

CK1 isoforms also have key roles in the developmentally important Wnt and Hedgehog (Hh) signaling pathways. When Wnt is not bound to its receptor, CK1α is thought to phosphorylate β-catenin as part of its ...

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Selective casein kinase 1ε inhibitor

Chemical Name: 3-[(3-Chlorophenoxy)methyl]-1-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine hydrochloride
Purity: ≥98% (HPLC)
Selective casein kinase 1ε inhibitor

Potent CK1 inhibitor; also inhibits cyclin-dependent kinases

Chemical Name: 2-[[9-(1-Methylethyl)-6-[[3-(2-pyridinyl)phenyl]amino]-9H-purin-2-yl]amino]-1-butanol dihydrochloride
Purity: ≥98% (HPLC)
Potent CK1 inhibitor; also inhibits cyclin-dependent kinases

CK1 inhibitor

Chemical Name: N-(2-Aminoethyl)-5-chloro-8-isoquinolinesulfonamide dihydrochloride
Purity: ≥99% (HPLC)
CK1 inhibitor

Selective CK1 inhibitor. Also inhibits TGF-βRI

Chemical Name: 4-[4-(2,3-Dihydro-1,4-benzodioxin-6-yl)-5-(2-pyridinyl)-1H-imidazol-2-yl]benzamide
Purity: ≥98% (HPLC)
Selective CK1 inhibitor. Also inhibits TGF-βRI

Potent and selective CK1ε and CK1δ inhibitor

Chemical Name: 4-[1-Cyclohexyl-4-(4-fluorophenyl)-1H-imidazol-5-yl]-2-pyrimidinamine dihydrochloride
Purity: ≥98% (HPLC)
Potent and selective CK1ε and CK1δ inhibitor

Potent CK1δ/ε inhibitor

Chemical Name: 4-[4-(4-Fluorophenyl)-1-[1-(3-isoxazolylmethyl)-4-piperidinyl]-1H-imidazol-5-yl]-2-pyrimidinamine
Purity: ≥98% (HPLC)
Potent CK1δ/ε inhibitor

Potent and selective CK1α, CK1δ and CK1ε inhibitor

Chemical Name: 4-(1-((4-Fluoro-1-methylpiperidin-4-yl)methyl)-4-(5-fluoropyridin-2-yl)-1H-imidazol-5-yl)-1H-pyrrolo[2,3-b]pyridine
Purity: ≥98% (HPLC)
Potent and selective CK1α, CK1δ and CK1ε inhibitor

Potent p38 MAPK inhibitor; anti-inflammatory

Chemical Name: N-[4-[2-Ethyl-4-(3-methylphenyl)-5-thiazolyl]-2-pyridinyl]benzamide
Purity: ≥98% (HPLC)
Potent p38 MAPK inhibitor; anti-inflammatory

Potent and selective CK1α molecular glue Degrader

Chemical Name: 3-(5-(Benzo[d]isoxazol-3-ylamino)-1-oxoisoindolin-2-yl)piperidine-2,6-dione
Purity: ≥98% (HPLC)
Potent and selective CK1α molecular glue Degrader
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