TGF-beta Receptor Inhibitors Products
17 results for "TGF-beta Receptor Inhibitors" in Products
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TGF-beta Receptor Inhibitors Products
17 results for "TGF-beta Receptor Inhibitors" in Products
Potent, selective inhibitor of TGF-βRI, ALK4 and ALK7
Chemical Name : | 4-[4-(1,3-benzodioxol-5-yl)-5-(2-pyridinyl)-1H-imidazol-2-yl]benzamide |
Purity : | ≥99% (HPLC) |
SB 431542 synthesized to cGMP guidelines
Chemical Name : | 4-[4-(1,3-benzodioxol-5-yl)-5-(2-pyridinyl)-1H-imidazol-2-yl]benzamide |
Purity : | ≥99% |
Selective inhibitor of TGF-βRI, ALK4 and ALK7
Chemical Name : | 3-(6-Methyl-2-pyridinyl)-N-phenyl-4-(4-quinolinyl)-1H-pyrazole-1-carbothioamide |
Purity : | ≥98% (HPLC) |
Selective inhibitor of TGF-βRI
Alternate Names : | HTS 466284 |
Chemical Name : | 4-[3-(2-Pyridinyl)-1H-pyrazol-4-yl]-quinoline |
Purity : | ≥99% (HPLC) |
Potent and selective inhibitor of TGF-βRI
Alternate Names : | E-616452, SJN 2511, ALK5 Inhibitor II |
Chemical Name : | 2-(3-(6-Methylpyridine-2-yl)-1H-pyrazol-4-yl)-1,5-naphthyridine |
Purity : | ≥99% (HPLC) |
RepSox synthesized to Ancillary Material Grade
Alternate Names : | ALK5 Inhibitor II, SJN 2511, E-616452 |
Chemical Name : | 2-[3-(6-Methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,5-naphthyridine |
Purity : | ≥99% |
Selective CK1 inhibitor. Also inhibits TGF-βRI
Chemical Name : | 4-[4-(2,3-Dihydro-1,4-benzodioxin-6-yl)-5-(2-pyridinyl)-1H-imidazol-2-yl]benzamide |
Purity : | ≥99% (HPLC) |
Potent and selective inhibitor of TGF-βRI
Chemical Name : | 4-[2-Fluoro-5-[3-(6-methyl-2-pyridinyl)-1H-pyrazol-4-yl]phenyl]-1H-pyrazole-1-ethanol |
Purity : | ≥98% (HPLC) |
Potent and selective inhibitor of TGF-βRI
Chemical Name : | 4-[4-[3-(2-Pyridinyl)-1H-pyrazol-4-yl]-2-pyridinyl]-N-(tetrahydro-2H-pyran-4-yl)-benzamide |
Purity : | ≥98% (HPLC) |
Selective inhibitor of TGF-βRI, ALK4 and ALK7
Chemical Name : | 2-[4-(1,3-Benzodioxol-5-yl)-2-(1,1-dimethylethyl)-1H-imidazol-5-yl]-6-methyl-pyridine |
Purity : | ≥98% (HPLC) |
Selective inhibitor of TGF-βRI
Chemical Name : | 6-[2-(1,1-Dimethylethyl)-5-(6-methyl-2-pyridinyl)-1H-imidazol-4-yl]quinoxaline |
Purity : | ≥97% (HPLC) |
Potent TGF-βRI inhibitor
Chemical Name : | 4-[[4-[(2.6-Dimethyl-3-pyridinyl)oxy]-2-pyridinyl]amino]benzenesulfonamide |
Purity : | ≥98% (HPLC) |
Potent ATP-competitive TGF-βRI inhibitor
Chemical Name : | 2-(5-Chloro-2-fluorophenyl)-4-[(4-pyridyl)amino]pteridine |
Purity : | ≥98% (HPLC) |
Potent inhibitor of TGF-βRI
Chemical Name : | 4-[3-(6-Methyl-2-pyridinyl)-1H-pyrazol-4-yl]quinoline |
Purity : | ≥98% (HPLC) |
ALK4 and ALK5 (TGFβRI) inhibitor
Alternate Names : | LY 2157299 |
Chemical Name : | 4-[5,6-Dihydro-2-(6-methyl-2-pyridinyl)-4H-pyrrolo[1,2-b]pyrazol-3-yl]-6-quinolinecarboxamide |
Purity : | ≥98% (HPLC) |
Potent TGF-βRI inhibitor; orally bioavailable
Chemical Name : | 4-[4-(1,3-Benzodioxol-5-yl)-5-(6-methyl-2-pyridinyl)-1H-imidazol-2-yl]bicyclo[2.2.2]octane-1-carboxamide |
Purity : | ≥98% (HPLC) |
Potent and selective inhibitor of TGF-βRI
Chemical Name : | 3-[[5-(6-Methyl-2-pyridinyl)-4-(6-quinoxalinyl)-1H-imidazol-2-yl]methyl]benzamide |
Purity : | ≥98% (HPLC) |