PARP2: Small Molecules and Peptides
6 results for "PARP2 Small Molecules and Peptides" in Products
6 results for "PARP2 Small Molecules and Peptides" in Products
PARP2: Small Molecules and Peptides
Potent tankyrase inhibitor
| Alternate Names: | XAV939 Wnt Signaling Inhibitor |
| Chemical Name: | 3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one |
| Purity: | ≥98% (HPLC) |
Potent PARP inhibitor
| Chemical Name: | 4-[[3-[[4-(Cyclopropylcarbonyl)-1-piperazinyl]carbonyl]-4-fluorophenyl]methyl]-1(2H)-phthalazinone |
| Purity: | ≥98% (HPLC) |
PARP inhibitor
| Alternate Names: | CO-338 |
| Chemical Name: | 8-Fluoro-1,3,4,5-tetrahydro-2-[4-[(methylamino)methyl]phenyl]-6H-pyrrolo[4,3,2,ef][2]benzazepin-6-one (1S,4R)-7,7-dimethyl-2-oxobicyclo[2.2.1]heptane-1-methanesulfonic acid |
| Purity: | ≥98% (HPLC) |
PARP inhibitor; photoaffinity probe
| Chemical Name: | 3-(3-Butyn-1-yl)-N-[5-cyano-6-[4-[3-[(3,4-dihydro-4-oxo-1-phthalazinyl)methyl]benzoyl]-1-piperazinyl]-3-pyridinyl]-3H-diazirine-3-propanamide |
| Purity: | ≥95% (HPLC) |
High affinity PARP-1 and -2 inhibitor; orally bioavailable
| Alternate Names: | ABT-888 |
| Chemical Name: | 2-[(2R)-2-Methyl-2-pyrrolidinyl]-1H-benzimidazole-4-carboxamide dihydrochloride |
| Purity: | ≥98% (HPLC) |
Potent PARP inhibitor
| Chemical Name: | N-(5,6-Dihydro-6-oxo-2-phenanthridinyl)-2-acetamide hydrochloride |
| Purity: | ≥98% (HPLC) |