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9 results for "fgf-receptor-inhibitors&view=expanded" in Products

Potent FGFR and VEGFR inhibitor

Alternate Names:
PF-02969207,PNU-0290908
Chemical Name:
2-[(1,2-Dihydro-2-oxo-3H-indol-3-ylidene)methyl]-4-methyl-1H-pyrrole-3-propanoic acid
Purity:
≥95%
Potent FGFR and VEGFR inhibitor

FGFR1 and -3 inhibitor

Chemical Name:
N-[2-[[4-(Diethylamino)butyl]amino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]-N'-(1,1-dimethylethyl)urea
Purity:
≥98%
FGFR1 and -3 inhibitor

Potent VEGFR, PDGFR and FGFR inhibitor

Chemical Name:
Methyl (Z)-3-[[[4-(N-methyl-2-(4-methylpiperazin-1-yl)acetamido)phenyl)amino)(phenyl)methylene]-2-oxoindoline-6-carboxylate
Purity:
≥98%
Potent VEGFR, PDGFR and FGFR inhibitor

FGFR1 and -3 inhibitor

Chemical Name:
N-[2-[[4-(Diethylamino)butyl]amino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]-N'-(1,1-dimethylethyl)urea
Purity:
≥98%
FGFR1 and -3 inhibitor

Potent and selective FGFR inhibitor

Chemical Name:
rel-N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-4-[(3R,5S)-3,5-dimethyl-1-piperazinyl]benzamide
Purity:
≥98%
Potent and selective FGFR inhibitor

Potent Src inhibitor; also inhibits FGFR1, PDGFRβ and Wee1

Chemical Name:
6-(2,6-Dichlorophenyl)-2-[[4-[2-(diethylamino)ethoxy]phenyl]amino]-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one dihydrochloride
Purity:
≥98%
Potent Src inhibitor; also inhibits FGFR1, PDGFRβ and Wee1

Potent inhibitor of VEGFR, PDGFR and FGFR

Chemical Name:
4-[(4-Fluoro-2-methyl-1H-indol-5-yl)oxy]-6-methoxy-7-[3-(1-pyrrolidinyl)propoxy]quinazoline
Purity:
≥98%
Potent inhibitor of VEGFR, PDGFR and FGFR

Potent multi-kinase and pan-Bcr-Abl inhibitor

Alternate Names:
Ponatinib
Chemical Name:
3-(2-Imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N-[4-[(4-methyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-benzamide
Purity:
≥98%
Potent multi-kinase and pan-Bcr-Abl inhibitor

DUSP6 and DUSP1 inhibitor

Chemical Name:
3-(Cyclohexylamino)-2,3-dihydro-2-(phenylmethylene)-1H-inden-1-one
Purity:
≥98%
DUSP6 and DUSP1 inhibitor
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