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Checkpoint Control Kinase Inhibitors: Small Molecules and Peptides
16 results for "Checkpoint Control Kinase Inhibitors Small Molecules and Peptides" in Products
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Checkpoint Control Kinase Inhibitors: Small Molecules and Peptides
16 results for "Checkpoint Control Kinase Inhibitors Small Molecules and Peptides" in Products
Inhibitor of PI 3-kinase, mTOR and DNA-PK
| Chemical Name : | 3-[4-(4-Morpholinylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl]phenol hydrochloride |
| Purity : | ≥98% (HPLC) |
Selective DNA-PK inhibitor
| Chemical Name : | 2-(4-Morpholinyl)-4H-naphthol[1,2-b]pyran-4-one |
| Purity : | ≥98% (HPLC) |
Selective Chk1 inhibitor
| Alternate Names : | PF-0044736 |
| Chemical Name : | (R)-α-Amino-N-[5,6-dihydro-2-(1-methyl-1H-pyrazol-4-yl)-6-oxo-1H-pyrrolo[4,3,2-ef][2,3]benzodiazepin-8-yl]-cyclohexaneacetamide |
| Purity : | ≥99% (HPLC) |
Potent and selective DNA-PK inhibitor
| Alternate Names : | KU 57788 |
| Chemical Name : | 8-(4-Dibenzothienyl)-2-(4-morpholinyl)-4H-1-benzopyran-4-one |
| Purity : | ≥99% (HPLC) |
MRN-ATM pathway inhibitor
| Chemical Name : | Z-5-(4-Hydroxybenzylidene)-2-imino-1,3-thiazolidin-4-one |
| Purity : | ≥99% (HPLC) |
Cdk inhibitor; potently inhibits cdk9; also inhibits MK2
| Chemical Name : | 1,5,6,7-Tetrahydro-2-(4-pyridinyl)-4H-pyrrolo[3,2-c]pyridin-4-one hydrochloride |
| Purity : | ≥99% (HPLC) |
Chk1 inhibitor
| Chemical Name : | 9,10,11,12-Tetrahydro- 9,12-epoxy-1H-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-1,3(2H)-dione |
| Purity : | ≥98% (HPLC) |
Dual DNA-PK and PI 3-K inhibitor
| Chemical Name : | 4-Ethyl-N-[4-[2-(4-morpholinyl)-4-oxo-4H-1-benzopyran-8-yl]-1-dibenzothienyl]-1-piperazineacetamide |
| Purity : | ≥97% (HPLC) |
Potent and selective Mps1 kinase inhibitor
| Chemical Name : | 9-Cyclopentyl-2-[[2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-phenyl]amino]-7-methyl-7,9-dihydro-8H-purin-8-one |
| Purity : | ≥99% (HPLC) |
Selective Chk2 inhibitor
| Alternate Names : | DDUG |
| Chemical Name : | 2,2'-[Carbonylbis(imino-4,1-phenyleneethylidyne]bishydrazinecarboximidamide) bis(4-methylbenzenesulfonate) |
| Purity : | ≥98% (HPLC) |
Selective Mps1 kinase inhibitor
| Chemical Name : | 1-[3-Methoxy-4-[[4-[[2-[(1-methylethyl)sulfonyl]phenyl]amino]-1H-pyrrolo[2,3-b]pyridin-6-yl]amino]phenyl]-4-piperidinol dihydrochloride |
| Purity : | ≥98% (HPLC) |
Potent Src inhibitor; also inhibits FGFR1, PDGFRβ and Wee1
| Chemical Name : | 6-(2,6-Dichlorophenyl)-2-[[4-[2-(diethylamino)ethoxy]phenyl]amino]-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one dihydrochloride |
| Purity : | ≥99% (HPLC) |
Potent and selective inhibitor of Chk1 and Wee1
| Chemical Name : | 9-Hydroxy-4-phenyl-pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione |
| Purity : | ≥98% (HPLC) |
Potent and selective ATM kinase inhibitor
| Chemical Name : | 2-(4-Morpholinyl)-6-(1-thianthrenyl)-4H-pyran-4-one |
| Purity : | ≥98% (HPLC) |
Potent and selective BUB1 kinase inhibitor
| Chemical Name : | 2-[3,5-Difluoro-4-[[3-[5-methoxy-4-[(3-methoxy-4-pyridinyl)amino]-2-pyrimidinyl]-1H-indazol-1-yl]methyl]phenoxy]ethanol |
| Purity : | ≥98% (HPLC) |
Potent Chk1 inhibitor
| Chemical Name : | 4'-[5-[[3-[(Cyclopropylamino)methyl]phenyl]amino]-1H-pyrazol-3-yl]-[1,1'-biphenyl]-2,4-diol |
| Purity : | ≥97% (HPLC) |
