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12 results for "Checkpoint Control Kinase Inhibitors" in Products
Checkpoint Control Kinase Inhibitors
Potent and selective ATM kinase inhibitor
Chemical Name:
2-(4-Morpholinyl)-6-(1-thianthrenyl)-4H-pyran-4-one
Purity:
≥98%
Potent and selective DNA-PK inhibitor
Alternate Names:
KU 57788
Chemical Name:
8-(4-Dibenzothienyl)-2-(4-morpholinyl)-4H-1-benzopyran-4-one
Purity:
≥98%
Inhibitor of PI 3-kinase, mTOR and DNA-PK
Chemical Name:
3-[4-(4-Morpholinylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl]phenol hydrochloride
Purity:
≥97%
Chk1 inhibitor
Chemical Name:
9,10,11,12-Tetrahydro- 9,12-epoxy-1H-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-1,3(2H)-dione
Purity:
≥98%
Potent and selective inhibitor of Chk1 and Wee1
Chemical Name:
9-Hydroxy-4-phenyl-pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione
Purity:
≥98%
Potent Src inhibitor; also inhibits FGFR1, PDGFRβ and Wee1
Chemical Name:
6-(2,6-Dichlorophenyl)-2-[[4-[2-(diethylamino)ethoxy]phenyl]amino]-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one dihydrochloride
Purity:
≥98%
Potent and selective Mps1 kinase inhibitor
Chemical Name:
9-Cyclopentyl-2-[[2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-phenyl]amino]-7-methyl-7,9-dihydro-8H-purin-8-one
Purity:
≥98%
Cdk inhibitor; potently inhibits cdk9; also inhibits MK2
Chemical Name:
1,5,6,7-Tetrahydro-2-(4-pyridinyl)-4H-pyrrolo[3,2-c]pyridin-4-one hydrochloride
Purity:
≥98%
MRN-ATM pathway inhibitor
Chemical Name:
Z-5-(4-Hydroxybenzylidene)-2-imino-1,3-thiazolidin-4-one
Purity:
≥98%
Potent and selective BUB1 kinase inhibitor
Chemical Name:
2-[3,5-Difluoro-4-[[3-[5-methoxy-4-[(3-methoxy-4-pyridinyl)amino]-2-pyrimidinyl]-1H-indazol-1-yl]methyl]phenoxy]ethanol
Purity:
≥98%
Potent Src inhibitor; also inhibits FGFR1, PDGFRβ and Wee1
Chemical Name:
6-(2,6-Dichlorophenyl)-2-[[4-[2-(diethylamino)ethoxy]phenyl]amino]-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one dihydrochloride
Purity:
≥98%
Potent and selective CHK1 inhibitor
Chemical Name:
5-[[5-[2-[[(1R,2R)-2-Aminocyclobutyl]oxy]-6-methoxyphenyl]-1H-pyrazol-3-yl]amino]-2-pyrazinecarbonitrile formate
Purity:
≥98%