
Adenosine A1 Receptor Antagonists: Small Molecules and Peptides
Adenosine A1 Receptor (ADORA1) is an adenosine receptor that belongs to the G protein-coupled receptor 1 family. There are 3 types of adenosine receptors, each with a specific pattern of ligand binding and tissue distribution, and together they regulate a diverse set of physiologic functions. The ADORA1 receptor inhibits adenylyl cyclase, and plays a role in the fertilization process. Animal studies also suggest a role for A1 receptors in kidney function and ethanol intoxication.
4 results for "Adenosine A1 Receptor Antagonists Small Molecules and Peptides" in Products
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Adenosine A1 Receptor Antagonists: Small Molecules and Peptides
Adenosine A1 Receptor (ADORA1) is an adenosine receptor that belongs to the G protein-coupled receptor 1 family. There are 3 types of adenosine receptors, each with a specific pattern of ligand binding and tissue distribution, and together they regulate a diverse set of physiologic functions. The ADORA1 receptor inhibits adenylyl cyclase, and plays a role in the fertilization process. Animal studies also suggest a role for A1 receptors in kidney function and ethanol intoxication.
4 results for "Adenosine A1 Receptor Antagonists Small Molecules and Peptides" in Products
Selective A1 antagonist
Chemical Name : | 8-Cyclopentyl-1,3-dipropylxanthine |
Purity : | ≥99% (HPLC) |
Selective A1 antagonist
Alternate Names : | Rolofylline |
Chemical Name : | 8-(Hexahydro-2,5-methanopentalen-3a(1H)-yl)-3,7-dihydro-1,3-dipropyl-1H-purine-2,6-dione |
Purity : | ≥99% (HPLC) |
Potent and selective A1 antagonist
Chemical Name : | trans-4-[(2-Phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclohexanol |
Purity : | ≥99% (HPLC) |
High affinity adenosine A1 receptor antagonist
Alternate Names : | CPT, 8-Cyclopentyltheophylline |
Chemical Name : | 8-Cyclopentyltheophylline |
Purity : | ≥99% (HPLC) |