NK1 Receptor Antagonists: Small Molecules and Peptides
NK1R (Neurokinin-1 receptor), gene name TACR1 (tachykinin receptor-1), is a 100 kDa 7-transmembrane glycoprotein receptor for the proinflammatory tachykinin neuropeptide, substance P. NK1R is constitutively or inducibly expressed on a wide variety of cells, including monocytes, macrophages, microglia, lymphocytes, neutrophils, mast cells, and neurons.
13 results for "NK1 Receptor Antagonists Small Molecules and Peptides" in Products
13 results for "NK1 Receptor Antagonists Small Molecules and Peptides" in Products
NK1 Receptor Antagonists: Small Molecules and Peptides
NK1R (Neurokinin-1 receptor), gene name TACR1 (tachykinin receptor-1), is a 100 kDa 7-transmembrane glycoprotein receptor for the proinflammatory tachykinin neuropeptide, substance P. NK1R is constitutively or inducibly expressed on a wide variety of cells, including monocytes, macrophages, microglia, lymphocytes, neutrophils, mast cells, and neurons.
| Chemical Name: | 1-[2-[(3S)-3-(3,4-Dichlorophenyl)-1-[2-[3-(1-methylethoxy)phenyl]acetyl]-3-piperidinyl]ethyl]-4-phenyl-1-azoniabicyclo[2.2.2]octane chloride |
| Purity: | ≥97% (HPLC) |
| Chemical Name: | (2S,3S)-3-[[3,5-bis(Trifluoromethyl)phenyl]methoxy]-2-phenylpiperidine hydrochloride |
| Purity: | ≥98% (HPLC) |
| Chemical Name: | 5-[[(2R,3S)-2-[(1R)-1-[3,5-Bis(trifluoromethyl)phenyl]ethoxy]-3-(4-fluorophenyl)-4-morpholinyl]methyl]-1,2-dihydro-3H-1,2,4-triazol-3-one |
| Purity: | ≥98% (HPLC) |
| Chemical Name: | (4R)-4-Hydroxy-1-[(1-methyl-1H-indol-3-yl)carbonyl]-L-prolyl-N-methyl-3-(2-naphthalenyl)-N-(phenylmethyl)-L-alaninamide |
| Purity: | ≥98% (HPLC) |
| Chemical Name: | 3-(2,3-Difluoro-4-methoxyphenyl)-2,5-dimethyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
| Purity: | ≥98% (HPLC) |
| Chemical Name: | (2S,3S)-N-(2-Methoxyphenyl)methyl-2-diphenylmethyl-1-azabicyclo[2.2.2]octan-3-amine |
| Purity: | ≥98% (HPLC) |
| Chemical Name: | (2S,3S)-N-[(2-Methoxyphenyl)methyl]-2-phenyl-3-piperidinamine dihydrochloride |
| Purity: | ≥98% (HPLC) |
| Chemical Name: | (3aR,7aR)-Octahydro-2-[1-imino-2-(2-methoxyphenyl)ethyl]-7,7-diphenyl-4H-isoindol |
| Purity: | ≥97% (HPLC) |
| Chemical Name: | 1-[[(2-Nitrophenyl)amino]carbonyl]-L-prolyl-N-methyl-3-(2-naphthalenyl)-N-(phenylmethyl)-L-alaninamide |
| Purity: | ≥98% (HPLC) |
| Chemical Name: | (2S,3S)-N-[[2-Methoxy-5-(1H-tetrazol-1-yl)phenyl]methyl]-2-phenyl-3-piperidinamine dihydrochloride |
| Purity: | ≥98% (HPLC) |
| Chemical Name: | (2S,3S)-N-[[2-Methoxy-5-(trifluoromethoxy)phenyl]methyl]-2-phenyl-3-piperidinamine dihydrochloride |
| Purity: | ≥98% (HPLC) |
| Chemical Name: | 5-[[(2R,3S)-2-[(1R)-1-[3,5-Bis(trifluoromethyl)phenyl]ethoxy]-3-(4-fluorophenyl)-4-morpholinyl]methyl-N,N-dimethyl-1H-1,2,3-triazole-4-methanamine hydrochloride |
| Purity: | ≥98% (HPLC) |
