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Histamine H3 Receptor Agonists: Small Molecules and Peptides

Histamine is a ubiquitous messenger molecule released from mast cells, enterochromaffin-like cells, and neurons. Its various actions are mediated by histamine receptors Histamine H1 R, Histamine H2 R, Histamine H3 R and Histamine H4 R. HRH3 encodes one of the histamine receptors (H3) which belongs to the family 1 of G protein-coupled receptors. Histamine H3 R is an integral membrane protein and can regulate neurotransmitter release. It can also increase voltage-dependent calcium current in smooth muscles and innervates the blood vessels and the heart in cardiovascular system.

7 results for "Histamine H3 Receptor Agonists Small Molecules and Peptides" in Products

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Histamine H3 Receptor Agonists: Small Molecules and Peptides

Histamine is a ubiquitous messenger molecule released from mast cells, enterochromaffin-like cells, and neurons. Its various actions are mediated by histamine receptors Histamine H1 R, Histamine H2 R, Histamine H3 R and Histamine H4 R. HRH3 encodes one of the histamine receptors (H3) which belongs to the family 1 of G protein-coupled receptors. Histamine H3 R is an integral membrane protein and can regulate neurotransmitter release. It can also increase voltage-dependent calcium current in smooth muscles and innervates the blood vessels and the heart in cardiovascular system.

7 results for "Histamine H3 Receptor Agonists Small Molecules and Peptides" in Products

Endogenous histamine receptor agonist

Standard H3 and H4 agonist (H3 > H4)

Potent, standard H3 agonist

Standard H3 agonist. Also H4 agonist

Potent H3 agonist, highly selective over H4

Non-selective H3 agonist

High affinity H3 ligand

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