Multidrug Transporter Inhibitors: Small Molecules and Peptides
10 results for "Multidrug Transporter Inhibitors Small Molecules and Peptides" in Products
10 results for "Multidrug Transporter Inhibitors Small Molecules and Peptides" in Products
Multidrug Transporter Inhibitors: Small Molecules and Peptides
Potent inhibitor of multidrug and toxin extrusion (MATE) transporters; also DHFR and STAT3 inhibitor
| Chemical Name: | 5-(4-Chlorophenyl)-6-ethyl-2,4-pyrimidinediamine |
| Purity: | ≥98% (HPLC) |
Potent and selective BCRP inhibitor
| Chemical Name: | (3S,6S,12aS)-1,2,3,4,6,7,12,12a-Octahydro-9-methoxy-6-(2-methylpropyl)-1,4-dioxopyrazino[1',2':1,6]pyrido[3,4-b]indole-3-propanoic acid 1,1-dimethylethyl ester |
| Purity: | ≥98% (HPLC) |
P-gp and BCRP inhibitor
| Alternate Names: | GF 120918 |
| Chemical Name: | N-[4-[2-(3,4-Dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)ethyl]phenyl]-9,10-dihydro-5-methoxy-9-oxo-4-acridinecarboxamide hydrochloride |
| Purity: | ≥98% (HPLC) |
MRP and OAT3 inhibitor
| Chemical Name: | 4-(Dipropylsulfamoyl)benzoic acid |
| Purity: | ≥98% (HPLC) |
Inhibitor of P-gp-mediated MDR
| Alternate Names: | Valspodar |
| Chemical Name: | 6-[(2S,4R,6E)-4-methyl-2-(methylamino)-3-oxo-6-octenoic acid]-7-L-valine-cyclosporin A |
| Purity: | ≥98% (HPLC) |
Potent P-glycoprotein (P-gp) inhibitor
| Chemical Name: | N-[2-[[[4-[2-(3,4-dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)ethyl]phenyl]amino]carbonyl]-4,5-dimethoxyphenyl]-3-quinolinecarbxamide dihydrochloride |
| Purity: | ≥98% (HPLC) |
Potent CysLT1 (LTD4) inverse agonist. Also MRP1 inhibitor
| Alternate Names: | L-660711 |
| Chemical Name: | 3-[[[3-[(1E)-2-(7-Chloro-2-quinolinyl)ethenyl]phenyl][[3-(dimethylamino)-3-oxopropyl]thio]methyl]thio]propanoic acid |
| Purity: | ≥98% (HPLC) |
Selective MRP4 inhibitor
| Chemical Name: | 5-[(2-Benzothiazolylthio)methyl]-2,4-dihydro-4-methyl-3H-1,2,4-triazole-3-thione |
| Purity: | ≥98% (HPLC) |
P-gp inhibitor
| Chemical Name: | 4-(3,4-Dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)-N-2[2-(3,4-dimethoxyphenyl)ethyl]-6,7-dimethoxy-2-quinazolinamine hydrochloride |
| Purity: | ≥98% (HPLC) |
Selective BCRP inhibitor
| Chemical Name: | N-[4-(2-Hydroxyethyl)phenyl]-2-[(4-nitrobenzoyl)amino]benzamide |
| Purity: | ≥98% (HPLC) |
