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5 results for "Histamine H4R Small Molecules and Peptides" in Products
Histamine H4R Small Molecules and Peptides
Histamine is a ubiquitous messenger molecule released from mast cells, enterochromaffin-like cells, and neurons. Its various actions are mediated by a family of histamine receptors, which are a subset of the G protein-coupled receptor superfamily. Histamine H4R is a histamine receptor that is predominantly expressed in hematopoietic cells. Histamine H4R is thought to play a role in inflammation and allergy reponses.
H3 antagonist; also H4 inverse agonist
Chemical Name:
N-Cyclohexyl-4-(imidazol-4-yl)-1-piperidinecarbothioamide
Purity:
≥98%
Selective H4 antagonist
Chemical Name:
1-[(5-Chloro-1H-indol-2-yl)carbonyl]-4-methylpiperazine
Purity:
≥98%
Selective H4 antagonist; orally active
Alternate Names:
VUF 6002
Chemical Name:
1-[(5-Chloro-1H-benzimidazol-2-yl)carbonyl]-4-methylpiperazine maleate
Purity:
≥98%
High affinity and selective 5-HT7 antagonist; orally bioavailable
Chemical Name:
6-Chloro-2a-[4-[4-(4-chlorophenyl)-3,6-dihydro-1(2H)-pyridinyl]butyl]-2a,3,4,5-tetrahydrobenz[cd]indol-2(1H)-one hydrochloride
Purity:
≥98%
Selective H4 antagonist; orally active
Alternate Names:
VUF 6002
Chemical Name:
1-[(5-Chloro-1H-benzimidazol-2-yl)carbonyl]-4-methylpiperazine maleate
Purity:
≥98%