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Histamine H3 Receptor Antagonists Products
Histamine is a ubiquitous messenger molecule released from mast cells, enterochromaffin-like cells, and neurons. Its various actions are mediated by histamine receptors Histamine H1 R, Histamine H2 R, Histamine H3 R and Histamine H4 R. HRH3 encodes one of the histamine receptors (H3) which belongs to the family 1 of G protein-coupled receptors. Histamine H3 R is an integral membrane protein and can regulate neurotransmitter release. It can also increase voltage-dependent calcium current in smooth muscles and innervates the blood vessels and the heart in cardiovascular system.
5 results for "Histamine H3 Receptor Antagonists" in Products
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Histamine H3 Receptor Antagonists Products
Histamine is a ubiquitous messenger molecule released from mast cells, enterochromaffin-like cells, and neurons. Its various actions are mediated by histamine receptors Histamine H1 R, Histamine H2 R, Histamine H3 R and Histamine H4 R. HRH3 encodes one of the histamine receptors (H3) which belongs to the family 1 of G protein-coupled receptors. Histamine H3 R is an integral membrane protein and can regulate neurotransmitter release. It can also increase voltage-dependent calcium current in smooth muscles and innervates the blood vessels and the heart in cardiovascular system.
5 results for "Histamine H3 Receptor Antagonists" in Products
Highly potent H3 antagonist and H4 partial agonist
| Alternate Names : | VUF 9153 |
| Chemical Name : | N-(4-Chlorobenzyl)-S-[3-(4(5)-imidazolyl)propyl]isothiourea dihydrobromide |
| Purity : | ≥99% (HPLC) |
High affinity H3 antagonist
| Chemical Name : | 1-[3-[4-(1-Piperidinylmethyl)phenoxy]propyl]piperidine hydrochloride |
| Purity : | ≥99% (HPLC) |
Potent, selective H3 antagonist
| Chemical Name : | N-[2-(4-Iodophenyl)ethyl]-S-[3-(4(5)-imidazolyl)propyl]isothiourea dihydrobromide |
| Purity : | ≥98% (HPLC) |
H3 antagonist; also H4 inverse agonist
| Chemical Name : | N-Cyclohexyl-4-(imidazol-4-yl)-1-piperidinecarbothioamide |
| Purity : | ≥99% (HPLC) |
Selective H3 antagonist and inverse agonist; also σ1 receptor antagonist; antinociceptive
| Chemical Name : | rel-4-[3-[(3aR,6aS)-Hexahydrocyclopenta[c]pyrrol-2(1H)-yl]propoxy]benzamide |
| Purity : | ≥98% (HPLC) |
