Clobenpropit dihydrobromide

Tocris Bioscience, part of Bio-Techne | Catalog # 0752

Highly potent H3 antagonist and H4 partial agonist
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Key Product Details

Description

Highly potent H3 antagonist and H4 partial agonist

Alternative Names

VUF 9153

View all Histamine H3 Receptor Antagonists »

Product Description

An extremely potent histamine H3 antagonist/inverse agonist (pA2=9.93). Also displays partial agonist activity at H4 receptors; induces eosinophil shape change with an EC50 of 3 nM.

Licensing Information

Sold with the permission of SCI, Amsterdam

Product Specifications

Molecular Weight

470.65

Formula

C14H17ClN4S.2HBr

Storage

Store at RT

Purity

≥98% (HPLC)

Chemical Name

N-(4-Chlorobenzyl)-S-[3-(4(5)-imidazolyl)propyl]isothiourea dihydrobromide

CAS Number

145231-35-2

PubChem ID

11213569

InChI Key

JIJQPEZAVLJZBO-UHFFFAOYSA-N

SMILES

Br.Br.ClC1=CC=C(CNC(=N)SCCCC2=CNC=N2)C=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 100

Preparing Stock Solutions for Clobenpropit dihydrobromide

The following data is based on the product molecular weight 470.65

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.12 mL 10.62 mL 21.25 mL
5 mM 0.42 mL 2.12 mL 4.25 mL
10 mM 0.21 mL 1.06 mL 2.12 mL
50 mM 0.04 mL 0.21 mL 0.42 mL

Calculators

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Background References

References are publications that support the biological activity of the product.

Product Documents for Clobenpropit dihydrobromide

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Clobenpropit dihydrobromide

For research use only

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