ZM 241385

Citations are publications that use Bio-Techne products. Selected citations for ZM 241385 include:

• Ryzhov et al. (2019) Number of Circulating CD 73-Expressing Lymphocytes Correlates With Survival After Cardiac Arrest. J Am Heart Assoc. 8:e010874
  PMID: 31237169
• Nuccio et al. (2019) Adenosine A2A receptor stimulation restores cell functions and differentiation in Niemann-Pick type C-like oligodendrocytes. Sci Rep. 9:9782
  PMID: 31278313
• Hirata et al. (2018) CD150high Bone Marrow Tregs Maintain Hematopoietic Stem Cell Quiescence and Immune Privilege via Adenosine. Cell Stem Cell. 22:445
  PMID: 29456159
• Ng (2018) Inhibition of cytokine-mediated JNK signalling by purinergic P2Y11 receptors, a novel protective mechanism in endothelial cells. Cell Signal. 51:59
  PMID: 30076967
• Wakisaka et al. (2017) An Adenosine Receptor for Olfaction in Fish. Curr Biol. 27:1437
  PMID: 28502661
• Liu et al. (2016) Activation of Adenosine 2A receptor inhibits neutrophil apoptosis in an autophagy-dependent manner in mice with systemic inflammatory response syndrome. Scientific Reports. 6:33614
  PMID: 27647162
• Mediero et al. (2016) Ticagrelor regulates osteoblast and osteoclast function and promotes bone formation in vivo via an adenosine-dependent mechanism. FASEB J.. 2016;
  PMID: 27511945
• Caiazzo et al. (2016) Adenosine signalling mediates the anti-inflammatory effects of the COX-2 inhibitor nimesulide. Biochem.Pharmacol.. 112:72
  PMID: 27188793
• Stoddart et al. (2015) Application of BRET to monitor ligand binding to GPCRs. Nat Methods. 12:661
  PMID: 26030448
• Hegde et al. (2015) Critical Role of Mast Cells and Peroxisome Proliferator-Activated Receptor γ in the Induction of Myeloid-Derived Suppressor Cells by Marijuana Cannabidiol In Vivo. J Immunol. 194:5211
  PMID: 25917103
• Cunha et al. (2015) Creatine, similarly to KA, affords antidepressant-like effects in the tail suspension test via adenosine A1 and A2A receptor activation. Biochem J. 11:215
  PMID: 25702084
• Tosolini et al. (2015) Human monocyte recognition of adenosine-based cyclic dinucleotides unveils the A2a Gαs protein-coupled receptor tonic inhibition of mitochondrially induced cell death. Am J Physiol Lung Cell Mol Physiol. 35:479
  PMID: 25384972
• Jamshad et al. (2015) G-protein coupled receptor solubilization and purification for biophysical analysis and functional studies, in the total absence of detergent. Mol Cell Biol. 35
  PMID: 25720391
• Kohno et al. (2015) Anti-inflammatory effects of adenosine N1-oxide. Biosci Rep. 12:2
  PMID: 25632271
• Oliveira et al. (2015) Deficits in endogenous adenosine formation by ecto-5'-nucleotidase/CD73 impair neuromuscular transmission and immune competence in experimental autoimmune myasthenia gravis. Mediators Inflamm. 2015:460610
  PMID: 25691808
• Perez-Aso et al. (2015) Apremilast, a novel phosphodiesterase 4 (PDE4) inhibitor, regulates inflammation through multiple cAMP downstream effectors. Arthritis Res Ther. 17:249
  PMID: 26370839
• Perígolo-Vicente et al. (2014) IL-6, A1 and A2aR: a crosstalk that modulates BDNF and induces neuroprotection. Biochem Biophys Res Commun. 449:477
  PMID: 24845382
• Ruby et al. (2014) Adenosinergic regulation of striatal clock gene expression and ethanol intake during constant light. Kidney Int. 39:2432
  PMID: 24755889
• Welihinda and Amento et al. (2014) Positive allosteric modulation of the adenosine A2a receptor attenuates inflammation. J Inflamm (Lond). 11:37
  PMID: 25473378
• Chiodi et al. (2014) Cocaine-induced changes of synaptic transmission in the striatum are modulated by adenosine A2A receptors and involve the tyrosine phosphatase STEP. Neuropsychopharmacology. 39:569
  PMID: 23989619
• Ahsan and Mehal (2014) Activation of adenosine receptor A2A increases HSC proliferation and inhibits death and senescence by down-regulation of p53 and Rb. Front Pharmacol. 5:69
  PMID: 24782773
• Sassi et al. (2014) Cardiac myocyte-secreted cAMP exerts paracrine action via adenosine receptor activation. J Clin Invest. 124:5385
  PMID: 25401477
• Mediavilla-Varela et al. (2013) Antagonism of adenosine A2A receptor expressed by lung adenocarcinoma tumor cells and cancer associated fibroblasts inhibits their growth. Neuropsychopharmacology. 14:860
  PMID: 23917542
• Hein et al. (2013) Cellular signalling pathways mediating dilation of porcine pial arterioles to adenosine A2A receptor activation. Blood. 99:156
  PMID: 23539502
• Nam et al. (2013) Adenosine transporter ENT1 regulates the acquisition of goal-directed behavior and ethanol drinking through A2A receptor in the dorsomedial striatum. J Neurosci. 33:4329
  PMID: 23467349
• Jenabian et al. (2013) Regulatory T cells negatively affect IL-2 production of effector T cells through CD39/adenosine pathway in HIV infection. PLoS Pathog. 9:e1003319
  PMID: 23658513
• Fernández-Dueñas et al. (2013) DA D(2) receptor-mediated modulation of adenosine A(2A) receptor agonist binding within the A(2A)R/D(2)R oligomer framework. Oncoimmunology. 63:42
  PMID: 23619397
• Jastrzebska et al. (2013) Expression of mammalian G protein-coupled receptors in Caenorhabditis elegans. J Neurochem. 520:239
  PMID: 23332703
• He et al. (2013) Adenosine regulates bone metabolism via A1, A2A, and A2B receptors in bone marrow cells from normal humans and patients with multiple myeloma. FASEB J. 27:3446
  PMID: 23682121
• Mandapathil et al. (2012) CD26 expression and adenosine deaminase activity in regulatory T cells (Treg) and CD4(+) T effector cells in patients with head and neck squamous cell carcinoma. FASEB J. 1:659
  PMID: 22934258
• Tozzi et al. (2012) A2A adenosine receptor antagonism enhances synaptic and motor effects of cocaine via CB1 cannabinoid receptor activation. PLoS One. 7:e38312
  PMID: 22715379
• Jeon et al. (2012) Oroxylin A Induces BDNF Expression on Cortical Neurons through Adenosine A2A Receptor Stimulation: A Possible Role in Neuroprotection. Neurochem Int. 20:27
  PMID: 24116271
• Lee et al. (2012) Polyphenol (-)-epigallocatechin gallate-induced cardioprotection may attenuate ischemia-reperfusion injury through adenosine receptor activation: a preliminary study. Biomol Ther (Seoul). 63:340
  PMID: 23115687
• Williams and Cronstein (2012) The effect of A(2A) adenosine receptor activation on C-C chemokine receptor 7 expression in human THP1 macrophages during inflammation. Inflammation. 35:614
  PMID: 21739164
• Lee et al. (2012) When cytokinin, a plant hormone, meets the adenosine A2A receptor: a novel neuroprotectant and lead for treating neurodegenerative disorders? PLoS One. 7:e38865
  PMID: 22719969
• Suzuki et al. (2012) CD8+CD45RA+CCR7+FOXP3+ T cells with immunosuppressive properties: a novel subset of inducible human regulatory T cells. J Immunol. 189:2118
  PMID: 22821963
• Fernández-Dueñas et al. (2012) Molecular determinants of A2AR-D2R allosterism: role of the intracellular loop 3 of the D2R. Invest Ophthalmol Vis Sci. 123:373
  PMID: 22924752
• Kinsey et al. (2012) Autocrine adenosine signaling promotes regulatory T cell-mediated renal protection. J Am Soc Nephrol. 23:1528
  PMID: 22835488
• Golembiowska and Dziubina (2012) The effect of adenosine A(2A) receptor antagonists on hydroxyl radical, DA, and glutamate in the striatum of rats with altered function of VMAT2. Neurotox Res. 22:150
  PMID: 22407500
• Waickman et al. (2012) Enhancement of tumor immunotherapy by deletion of the A2A adenosine receptor. Cancer Immunol Immunother. 61:917
  PMID: 22116345
• Takedachi et al. (2012) CD73-generated adenosine promotes osteoblast differentiation. J Cell Physiol. 227:2622
  PMID: 21882189
• Lindquist (2012) Adenosine receptor activation is responsible for prolonged depression of synaptic transmission after spreading depolarization in brain slices. Neuroscience. 223:365
  PMID: 22864185
• Stoddart et al. (2012) Fragment screening at adenosine-A(3) receptors in living cells using a fluorescence-based binding assay. Chem Biol. 19:1105
  PMID: 22999879
• Mediero et al. (2012) Adenosine A2A receptor activation prevents wear particle-induced osteolysis. Sci Transl Med. 4:135ra65
  PMID: 22623741
• Kiebala and Maggirwar (2011) Ibudilast, a pharmacologic phosphodiesterase inhibitor, prevents human immunodeficiency virus-1 Tat-mediated activation of microglial cells. PLoS One. 6:e18633
  PMID: 21494611
• Jin et al. (2011) Paeoniflorin suppresses the expression of intercellular adhesion molecule-1 (ICAM-1) in endotoxin-treated human monocytic cells. Br J Pharmacol. 164:694
  PMID: 21542832
• Tozzi et al. (2011) The distinct role of medium spiny neurons and cholinergic interneurons in the D2/A2A receptor interaction in the striatum: implications for Parkinson's disease. J Neurosci. 31:1850
  PMID: 21289195
• Garcia et al. (2011) Adenosine A(2A) receptor activation prevents progressive kidney fibrosis in a model of immune-associated chronic inflammation. Proc Natl Acad Sci U S A. 80:378
  PMID: 21508927
• Ruiz-García et al. (2011) Cooperation of adenosine with macrophage Toll-4 receptor agonists leads to increased glycolytic flux through the enhanced expression of PFKFB3 gene. J Biol Chem. 286:19247
  PMID: 21464136
• Zhukov et al. (2011) Biophysical mapping of the adenosine A2A receptor. J Med Chem. 54:4312
  PMID: 21661720
• Gebremedhin et al. (2010) Adenosine can mediate its actions through generation of reactive oxygen species. J Cereb Blood Flow Metab. 30:1777
  PMID: 20531463
• Himer et al. (2010) Adenosine A2A receptor activation protects CD4+ T lymphocytes against activation-induced cell death. FASEB J. 24:2631
  PMID: 20371613
• Gazoni et al. (2010) Activation of A1, A2A, or A3 adenosine receptors attenuates lung ischemia-reperfusion injury. J Thorac Cardiovasc Surg. 140:440
  PMID: 20398911
• Bingham et al. (2010) A2A adenosine receptor stimulation decreases foam cell formation by enhancing ABCA1-dependent cholesterol efflux. J Leukoc Biol. 87:683
  PMID: 20089670
• Nowak et al. (2010) The A2aR adenosine receptor controls cytokine production in iNKT cells. Am J Pathol. 40:682
  PMID: 20039304
• Long et al. (2010) Adenosine receptor regulation of coronary blood flow in Ossabaw miniature swine. J Exp Med. 335:781
  PMID: 20855445
• Paisansathan et al. (2010) Interactions between adenosine and K+ channel-related pathways in the coupling of somatosensory activation and pial arteriolar dilation. Am J Physiol Heart Circ Physiol. 299:H2009
  PMID: 20889844
• Wang et al. (2010) Static magnetic field exposure reproduces cellular effects of the Parkinson's disease drug candidate ZM241385. Korean J Anesthesiol. 5:e13883
  PMID: 21079735
• Riccioni et al. (2010) Adenosine A(2A) Receptor Binding Profile of Two Antagonists, ST1535 and KW6002: Consideration on the Presence of Atypical Adenosine A(2A) Binding Sites. Front Psychiatry. 1:22
  PMID: 21423433
• Carlström et al. (2010) Adenosine A(2) receptors modulate tubuloglomerular feedback. Am J Physiol Renal Physiol. 299:F412
  PMID: 20519378
• Mandapathil et al. (2010) Generation and accumulation of immunosuppressive adenosine by human CD4+CD25highFOXP3+ regulatory T cells. J Biol Chem. 285:7176
  PMID: 19858205
• Pugliese et al. (2009) The adenosine A2A receptor antagonist ZM241385 enhances neuronal survival after oxygen-glucose deprivation in rat CA1 hippocampal slices. Br J Pharmacol. 157:818
  PMID: 19422385
• Epperson et al. (2009) Adenosine receptors and second messenger signaling pathways in rat cardiac fibroblasts. Am J Physiol Cell Physiol. 296:C1171
  PMID: 19244482
• Clark et al. (2009) Adenosine-evoked hyperpolarization of retinal ganglion cells is mediated by G-protein-coupled inwardly rectifying K+ and small conductance Ca²⁺-activated K+ channel activation. J Neurosci. 29:11237
  PMID: 19741130
• Alam et al. (2009) A2A adenosine receptor (AR) activation inhibits pro-inflammatory cytokine production by human CD4+ helper T cells and regulates Helicobacter-induced gastritis and bacterial persistence. Mucosal Immunol. 2:232
  PMID: 19262506
• Yu et al. (2009) Effect of ventilation pressure on alveolar fluid clearance and β-agonist responses in mice. Cancer Biol Ther. 297:L785
  PMID: 19684202
• Ohta et al. (2009) A2A adenosine receptor may allow expansion of T cells lacking effector functions in extracellular adenosine-rich microenvironments. Cardiovasc Res. 183:5487
  PMID: 19843934
• Wilson et al. (2009) The A2B adenosine receptor impairs the maturation and immunogenicity of dendritic cells. J Immunol. 182:4616
  PMID: 19342636
• Maeda and Koos (2009) Adenosine A1 and A2a receptors modulate Insemia, glycemia, and lactatemia in fetal sheep. Proc Natl Acad Sci U S A. 296:R693
  PMID: 19118101
• Shi et al. (2008) Interaction of mechanisms involving epoxyeicosatrienoic acids, adenosine receptors, and metabotropic glutamate receptors in neurovascular coupling in rat whisker barrel cortex. J Cereb Blood Flow Metab. 28:111
  PMID: 17519974
• Csóka et al. (2008) Adenosine A2A receptor activation inhibits T helper 1 and T helper 2 cell development and effector function. FASEB J. 22:3491
  PMID: 18625677
• Fernandez et al. (2008) Pharmacological blockade of A2A receptors prevents dermal fibrosis in a model of elevated tissue adenosine. J Pharmacol Exp Ther. 172:1675
  PMID: 18467695
• Garcia et al. (2008) Adenosine A2A receptor activation and macrophage-mediated experimental glomerulonephritis. Am J Physiol Regul Integr Comp Physiol. 22:445
  PMID: 17898087
• Singh et al. (2008) Large-scale functional expression of WT and truncated human adenosine A2A receptor in Pichia pastoris bioreactor cultures. Eur J Immunol. 7:28
  PMID: 18847468
• Liou et al. (2008) Mediation of cannabidiol anti-inflammation in the retina by equilibrative nucleoside transporter and A2A adenosine receptor. PLoS One. 49:5526
  PMID: 18641283
• Ramanathan et al. (2007) Synergistic up-regulation of vascular endothelial growth factor (VEGF) expression in macrophages by adenosine A2A receptor agonists and endotoxin involves transcriptional regulation via the hypoxia response element in the VEGF promoter. Br J Pharmacol. 18:14
  PMID: 17065555
• Chan et al. (2006) Adenosine A(2A) receptors play a role in the pathogenesis of hepatic cirrhosis. Br J Pharmacol. 148:1144
  PMID: 16783407
• Zhang et al. (2006) Adenosine A2a receptors induce heterologous desensitization of chemokine receptors. Microb Cell Fact. 108:38
  PMID: 16522819
• Ge et al. (2006) Cl-IB-MECA [2-chloro-N6-(3-iodobenzyl)adenosine-5'-N-methylcarboxamide] reduces ischemia/reperfusion injury in mice by activating the A3 adenosine receptor. J Inflamm (Lond). 319:1200
  PMID: 16985166
• Lappas et al. (2006) Adenosine A2A receptor activation reduces hepatic ischemia reperfusion injury by inhibiting CD1d-dependent NKT cell activation. Mol Biol Cell. 203:2639
  PMID: 17088433
• Bertarelli et al. (2006) Characterization of human and rodent native and recombinant adenosine A(2B) receptors by radioligand binding studies. Purinergic Signal. 2:559
  PMID: 18404493
• Jacobson et al. (2005) A neoceptor approach to unraveling microscopic interactions between the human A2A adenosine receptor and its agonists. Chem Biol. 12:237
  PMID: 15734651
• Murphree et al. (2005) Lipopolysaccharide rapidly modifies adenosine receptor transcripts in murine and human macrophages: role of NF-κB in A(2A) adenosine receptor induction. Methods Enzymol. 391:575
  PMID: 16022683
• Erdmann et al. (2005) Activation of Th1 and Tc1 cell adenosine A2A receptors directly inhibits IL-2 secretion in vitro and IL-2-driven expansion in vivo. J Pharmacol Exp Ther. 105:4707
  PMID: 15746085
• Kornerup et al. (2005) Pharmacological characterisation of the adenosine receptor mediating increased ion transport in the mouse isolated trachea and the effect of allergen challenge. Br J Pharmacol. 144:1011
  PMID: 15685200
• Newman (2005) Calcium increases in retinal glial cells evoked by light-induced neuronal activity. Blood. 25:5502
  PMID: 15944378
• Fresco et al. (2004) Facilitation of noradrenaline release by activation of adenosine A(2A) receptors triggers both phospholipase C and adenylate cyclase pathways in rat tail artery. Cardiovasc Res. 63:739
  PMID: 15306230
• Yip (2004) Role of adenosine A2A receptor in the regulation of gastric somatostatin release. J Pharmacol Exp Ther. 309:804
  PMID: 14742743
• Germack and Dickenson (2004) Characterization of ERK1/2 signalling pathways induced by adenosine receptor subtypes in newborn rat cardiomyocytes. Br J Pharmacol. 141:329
  PMID: 14751870
• Wen and Knowles (2003) Extracellular ATP and adenosine induce cell apoptosis of human hepatoma Li-7A cells via the A3 adenosine receptor. Br J Pharmacol. 140:1009
  PMID: 14530217
• Dall'Igna et al. (2003) Neuroprotection by caffeine and adenosine A2A receptor blockade of β-amyloid neurotoxicity. PLoS One. 138:1207
  PMID: 12711619
• Nishi et al. (2003) Metabotropic mGlu5 receptors regulate adenosine A2A receptor signaling. Br J Pharmacol. 100:1322
  PMID: 12538871
• Koshiba et al. (2002) 2-Chloroadenosine but not adenosine induces apoptosis in rheumatoid fibroblasts independently of cell surface adenosine receptor signalling. Br J Pharmacol. 135:1477
  PMID: 11906961
• Brito et al. (2002) Adenosine A(2A) receptors in portal hypertension: their role in the abnormal response to adenosine of the cranial mesenteric artery in rabbits. J Neurosci. 135:1324
  PMID: 11877342
• Hirsh and Silinsky (2002) Inhibition of spontaneous acetylcholine secretion by 2-chloroadenosine as revealed by a protein kinase inhibitor at the mouse neuromuscular junction. Br J Pharmacol. 135:1897
  PMID: 11959792
• Slesinger (2001) British Pharmacological Society Meeting. 18-21 December 2000, University of Birmingham. Abstracts. Br J Pharmacol. 133 Suppl:1P
  PMID: 11403025
• Avila et al. (2001) A(1)-, A(2A)- and A(3)-subtype adenosine receptors modulate intraocular pressure in the mouse. Br J Pharmacol. 134:241
  PMID: 11564641
• Nieri et al. (2001) Adenosine-mediated hypotension in in vivo guinea-pig: receptors involved and role of NO. Br J Pharmacol. 134:745
  PMID: 11606314
• Lee and Chao (2001) Activation of Trk neurotrophin receptors in the absence of neurotrophins. Purinergic Signal. 98:3555
  PMID: 11248116
• Anderson et al. (2000) Accelerated resequestration of cytosolic calcium and suppression of the pro-inflammatory activities of human neutrophils by CGS 21680 in vitro. Br J Pharmacol. 130:717
  PMID: 10864876
• Haynes (2000) A(2A) adenosine receptor mediated potassium channel activation in rat epididymal smooth muscle. Br J Pharmacol. 130:685
  PMID: 10821799
• Hernandez et al. (1999) A2B adenosine receptors mediate relaxation of the pig intravesical ureter: adenosine modulation of non adrenergic non cholinergic excitatory neurotransmission. Br J Pharmacol. 126:969
  PMID: 10193777
• Latini et al. (1999) Effect of A2A adenosine receptor stimulation and antagonism on synaptic depression induced by in vitro ischaemia in rat hippocampal slices. Br J Pharmacol. 128:1035
  PMID: 10556941
• Haynes et al. (1998) A1 and A2 adenosine receptor modulation of contractility in the cauda epididymis of the guinea-pig. Br J Pharmacol. 125:570
  PMID: 9806342
• Guibert et al. (1998) Dependence of P2-nucleotide receptor agonist-mediated endothelium-independent relaxation on ectonucleotidase activity and A2A-receptors in rat portal vein. Br J Pharmacol. 123:1732
  PMID: 9605582
• Nakav et al. Anti-inflammatory preconditioning by agonists of adenosine A1 receptor. J Immunol. 3:e2107
  PMID: 18461129

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• Mouse solenocytes

  Name: Tahmineh Safaie
  Species: Mouse
  Assay Type: Ex Vivo
  Cell Line/Tissue: solenocytes
  Mouse solenocytes were activated with antiCD3/28 and treated with 5 uM of ZM241385 in presence or absence of CGS21680. After 24 hours the supernatant was collected, and IFN-gamma was measured by ELISA.
  

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