Adenosine A2a Receptor Antagonists Products
Adenosine A2A Receptor (ADORA2A) is one of several receptor subtypes for adenosine. The activity of ADORA2A, a G protein-coupled receptor family member, is mediated by G proteins which activate adenylyl cyclase. ADORA2A is abundant in basal ganglia, vasculature and platelets and is a major target of caffeine. Variability in the acute blood pressure response to coffee may be partly explained by genetic polymorphisms of the adenosine A2A receptors, including ADORA2A, and alpha(2)-adrenergic receptors.
6 results for "Adenosine A2a Receptor Antagonists" in Products
6 results for "Adenosine A2a Receptor Antagonists" in Products
Adenosine A2a Receptor Antagonists Products
Adenosine A2A Receptor (ADORA2A) is one of several receptor subtypes for adenosine. The activity of ADORA2A, a G protein-coupled receptor family member, is mediated by G proteins which activate adenylyl cyclase. ADORA2A is abundant in basal ganglia, vasculature and platelets and is a major target of caffeine. Variability in the acute blood pressure response to coffee may be partly explained by genetic polymorphisms of the adenosine A2A receptors, including ADORA2A, and alpha(2)-adrenergic receptors.
Potent and highly selective A2A antagonist
| Chemical Name: | 4-(2-[7-Amino-2-(2-furyl)[1,2,4]triazolo[2,3-a][1,3,5]triazin-5-ylamino]ethyl)phenol |
| Purity: | ≥99% (HPLC) |
Potent, highly selective A2A antagonist
| Chemical Name: | 2-(2-Furanyl)-7-(2-phenylethyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine |
| Purity: | ≥99% (HPLC) |
Adenosine A2A antagonist
| Chemical Name: | 8-Ethoxy-9-ethyl-9H-purin-6-amine |
| Purity: | ≥99% (HPLC) |
Potent and selective A2A antagonist
| Alternate Names: | KW-6002 |
| Chemical Name: | 8-[(1E)-2-(2-(3,4-Dimethoxyphenyl)ethenyl]-1,3-diethyl-3,7-dihydro-7-methyl-1H-purine-2,6-dione |
| Purity: | ≥99% (HPLC) |
Very selective, high affinity A2A antagonist
| Chemical Name: | 2-(2-Furanyl)-7-[3-(4-methoxyphenyl)propyl]-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine |
| Purity: | ≥99% (HPLC) |
Potent and selective A2A antagonist
| Chemical Name: | N-[2-(3,5-Dimethyl-1H-pyrazol-1-yl)-6-[6-(4-methoxy-1-piperidinyl)-2-pyridinyl]-4-pyrimidinyl]acetamide |
| Purity: | ≥98% (HPLC) |
