Zaprinast

Tocris Bioscience, part of Bio-Techne | Catalog # 0947

GPR35 agonist
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Key Product Details

Description

GPR35 agonist

View all Phosphodiesterase Inhibitors »

Product Description

Zaprinast is a phosphodiesterase inhibitor, selective for PDE6, 5, 11 and 9 (IC50 values are 0.15, 0.76, 12.0 and 29.0 μM respectively). Putative GPR35 agonist.

Product Specifications

Molecular Weight

271.28

Formula

C13H13N5O2

Storage

Store at RT

Purity

≥98% (HPLC)

Chemical Name

2-(2-Propyloxyphenyl)-8-azapurin-6-one

CAS Number

37762-06-4

PubChem ID

5722

InChI Key

REZGGXNDEMKIQB-UHFFFAOYSA-N

SMILES

CCCOC1=C(C=CC=C1)C1=NC2=C(NN=N2)C(=O)N1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 100

Preparing Stock Solutions for Zaprinast

The following data is based on the product molecular weight 271.28

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 3.69 mL 18.43 mL 36.86 mL
5 mM 0.74 mL 3.69 mL 7.37 mL
10 mM 0.37 mL 1.84 mL 3.69 mL
50 mM 0.07 mL 0.37 mL 0.74 mL

Calculators

Molarity Calculator

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Dilution Calculator

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Reconstitution Calculator

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Background References

References are publications that support the biological activity of the product.

Product Documents for Zaprinast

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Zaprinast

For research use only

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