2 results for "Kappa Opioid Receptor Antagonists Small Molecules and Peptides" in Products
Kappa Opioid Receptor Antagonists: Small Molecules and Peptides
The κ opioid receptor, (also known as OP2, KOP, KOR), is a member of the opioid family of G-protein-coupled receptors that also includes μ, δ and NOP receptors. Three variants of the receptor (designated κ1, κ2, and κ3) have been characterized. However only one cDNA clone has been identified, hence these receptor subtypes are likely to arise from interaction of one κ-opioid receptor protein with other membrane associated proteins.
κ Opioid receptors are ...
Selective κ opioid receptor antagonist
| Chemical Name: | N-[3-[4-(4-Methoxyphenyl)-1-piperazinyl]propyl]-1-methyl-6-oxopyrido[2,3-e]pyrrolo[1,2-a]pyrazine-5(6H)-acetamide |
| Purity: | ≥98% (HPLC) |
Selective and irreversible κ antagonist
| Chemical Name: | 2-(3,4-Dichlorophenyl)-N-methyl-N-[(1S)-1-(3-isothiocyanatophenyl)-2-(1-pyrrolidinyl)ethyl]acetamide hydrochloride |
| Purity: | ≥98% (HPLC) |
