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EZH2 Inhibitor: Small Molecules and Peptides
9 results for "EZH2 Inhibitor Small Molecules and Peptides" in Products
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EZH2 Inhibitor: Small Molecules and Peptides
9 results for "EZH2 Inhibitor Small Molecules and Peptides" in Products
EZH2 histone methyltransferase inhibitor
| Alternate Names : | DZNep, NSC 617989 |
| Chemical Name : | (1S,2R,5R)-5-(4-Amino-1H-imidazo[4,5-c]pyridin-1-yl)-3-(hydroxymethyl)-3-cyclopentene-1,2-diol hydrochloride |
| Purity : | ≥98% (HPLC) |
Catalog #:
TB4703-RMU
3-Deazaneplanocin A hydrochloride synthesized to Ancillary Material Grade
| Chemical Name : | (1S,2R,5R)-5-(4-Amino-1H-imidazo[4,5-c]pyridin-1-yl)-3-(hydroxymethyl)-3-cyclopentene-1,2-diol hydrochloride |
| Purity : | ≥98% |
Catalog #:
5847
Potent and selective EZH2 inhibitor; orally bioavailable
| Chemical Name : | 3-[Ethyl(tetrahydro-2H-pyran-4-yl)amino]-N-[(2,3,5,6,7,8-hexahydro-1-methyl-3-oxo-4-isoquinolinyl)methyl]-2-methyl-5-[6-(4-methyl-1-piperazinyl)-3-pyridinyl]benzamide |
| Purity : | ≥98% (HPLC) |
Catalog #:
6790
Very high affinity and selective EZH2 inhibitor
| Chemical Name : | N-[(1,2-Dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-3-methyl-1-[(1S)-1-methylpropyl]-6-[6-(1-piperazinyl)-3-pyridinyl]-1H-indole-4-carboxamide |
| Purity : | ≥98% (HPLC) |
Catalog #:
6153
Potent and selective SAM-competitive EZH2 inhibitor
| Chemical Name : | N-[(1,2-Dihydro-6-methyl-2-oxo-4-propyl-3-pyridinyl)methyl]-1-(1-methylethyl)-6-[6-(4-methyl-1-piperazinyl)-3-pyridinyl]-1H-pyrazolo[3,4-b]pyridine-4-carboxamide |
| Purity : | ≥98% (HPLC) |
Biotinylated UNC 1999 (Cat.No. 4904)
| Chemical Name : | 1-Isopropyl-N-[(6-methyl-2-oxo-4-propyl-1,2-dihydropyridin-3-yl)methyl]-6-[6-[4-[41-oxo-45-[(3aS,4aS,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl]-4,7,10,13,16,19,22,25,28,31,34,37-dodecaoxa-40-azapentatetracontan-1oyl]piperazin-1-yl]pyridin-3-yl]-1H-indazole-4-carboxamide |
| Purity : | ≥95% (HPLC) |
Potent and selective EZH2/EZH1 inhibitor
| Chemical Name : | N-[(1,2-Dihydro-6-methyl-2-oxo-4-propyl-3-pyridinyl)methyl]-1-(1-methylethyl)-6-[6-[4-(1-methylethyl)-1-piperazinyl]-3-pyridinyl]-1H-indazole-4-carboxamide |
| Purity : | ≥99% (HPLC) |
Catalog #:
6128
Potent and selective SAM-competitive EZH2 inhibitor
| Chemical Name : | N-[(1,2-Dihydro-6-methyl-2-oxo-4-propyl-3-pyridinyl)methyl]-1-(1-methylethyl)-6-[2-(4-methyl-1-piperazinyl)-4-pyridinyl]-1H-indazole-4-carboxamide |
| Purity : | ≥98% (HPLC) |
Catalog #:
6169
Highly potent and SAM-competitive EZH2 inhibitor
| Chemical Name : | 5,8-Dichloro-2-[(1,2-dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-7-(3,5-dimethyl-4-isoxazolyl)-3,4-dihydro-1(2H)-isoquinolinone acetate |
| Purity : | ≥97% (HPLC) |
