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5-HT1B Receptor Antagonists: Small Molecules and Peptides

5-HT1B is a 7TM receptor for serotonin and is expressed on striatal neurons and Purkinje cells in the cerebellum. 5-HT1B ligation inhibits glycinergic signaling, appetite, circadian rhythym light responsiveness, and trigeminal-mediated nociception. It is an important pharmacologic target in the treatment of migrane headaches.

7 results for "5-HT1B Receptor Antagonists Small Molecules and Peptides" in Products

5-HT1B Receptor Antagonists: Small Molecules and Peptides

5-HT1B is a 7TM receptor for serotonin and is expressed on striatal neurons and Purkinje cells in the cerebellum. 5-HT1B ligation inhibits glycinergic signaling, appetite, circadian rhythym light responsiveness, and trigeminal-mediated nociception. It is an important pharmacologic target in the treatment of migrane headaches.

7 results for "5-HT1B Receptor Antagonists Small Molecules and Peptides" in Products

β3 partial agonist; also 5-HT1A and 5-HT1B antagonist; more active enantiomer of pindolol (Cat. No. 0994)

Selective h5-HT1B antagonist

Selective 5-HT1B antagonist

Selective r5-HT1B antagonist; active in vivo

Potent and selective 5-HT1B and 5-HT1D antagonist

5-HT1B antagonist

5-HT1A and 5-HT1B antagonist; also β-adrenergic antagonist

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