Zacopride hydrochloride

Tocris Bioscience, part of Bio-Techne | Catalog # 1795

Highly potent 5-HT3 antagonist; also 5-HT4 agonist
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Key Product Details

Description

Highly potent 5-HT3 antagonist; also 5-HT4 agonist

View all 5-HT3 Receptor Antagonists »

Product Description

Zacopride hydrochloride is a highly potent 5-HT3 receptor antagonist (Ki = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). Antiemetic and anxiolytic following systemic administration in vivo.

Product Specifications

Molecular Weight

346.26

Formula

C15H20ClN3O2.HCl

Storage

Desiccate at RT

Purity

≥98% (HPLC)

Chemical Name

(±)-4-Amino-N-1-azabicyclo[2.2.2]oct-3-yl-5-chloro-2-methoxybenzamide hydrochloride

CAS Number

101303-98-4

PubChem ID

9928181

InChI Key

ITXVOUSORXSTQH-UHFFFAOYSA-N

SMILES

Cl.COC1=C(C=C(Cl)C(N)=C1)C(=O)NC1CN2CCC1CC2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 34.63 100
DMSO 34.62 100

Preparing Stock Solutions for Zacopride hydrochloride

The following data is based on the product molecular weight 346.26

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.89 mL 14.44 mL 28.88 mL
5 mM 0.58 mL 2.89 mL 5.78 mL
10 mM 0.29 mL 1.44 mL 2.89 mL
50 mM 0.06 mL 0.29 mL 0.58 mL

Calculators

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Background References

References are publications that support the biological activity of the product.

Product Documents for Zacopride hydrochloride

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Zacopride hydrochloride

For research use only

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