Rilmenidine hemifumarate

Tocris Bioscience, part of Bio-Techne | Catalog # 0790

I1 ligand. Also α2 agonist
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Key Product Details

Description

I1 ligand. Also α2 agonist

View all Adrenergic alpha-2 Receptor Agonists »

Product Description

Rilmenidine hemifumarate is an I1-imidazoline binding site selective ligand and α2-adrenoceptor agonist. Possesses greater I1 vs α2 selectivity than the prototypical compound, clonidine. Also thought to enhance autophagy; shown to increase LC3-II levels in PC12 cells.

Product Specifications

Molecular Weight

238.29

Formula

C10H16N2O.½C4H4O4

Storage

Store at -20°C

Purity

≥98% (HPLC)

Chemical Name

2-[N-(Dicyclopropylmethyl)amino]oxazoline hemifumarate

CAS Number

207572-68-7

PubChem ID

45073450

InChI Key

LZFATBMLSYHRTC-WXXKFALUSA-N

SMILES

OC(=O)\C=C\C(O)=O.C1CC1C(NC1=NCCO1)C1CC1.C1CC1C(NC1=NCCO1)C1CC1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 5.96 25

Preparing Stock Solutions for Rilmenidine hemifumarate

The following data is based on the product molecular weight 238.29

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.25 mM 16.79 mL 83.93 mL 167.86 mL
1.25 mM 3.36 mL 16.79 mL 33.57 mL
2.5 mM 1.68 mL 8.39 mL 16.79 mL
12.5 mM 0.34 mL 1.68 mL 3.36 mL

Calculators

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Background References

References are publications that support the biological activity of the product.

Product Documents for Rilmenidine hemifumarate

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Rilmenidine hemifumarate

For research use only

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