PSB 0788
Tocris Bioscience, part of Bio-Techne | Catalog # 3199
Selective A2B antagonist
Key Product Details
Description
Selective A2B antagonist
Product Description
PSB 0788 is a potent and selective adenosine A2B receptor antagonist (IC50 = 3.64 nM at human A2B receptors). Displays > 100-fold selectivity over hA1, hA2A and hA3 receptors.Product Specifications
Molecular Weight
543.04
Formula
C25H27ClN6O4S
Storage
Store at +4°C
Purity
≥98% (HPLC)
Chemical Name
8-[4-[4-(4-Chlorobenzyl)piperazide-1-sulfonyl)phenyl]]-1-propylxanthine
CAS Number
1027513-54-7
PubChem ID
44186581
InChI Key
JQZJACVYMPKVDS-UHFFFAOYSA-N
SMILES
O=C(NC2=C1NC(C3=CC=C(S(N4CCN(CC5=CC=C(Cl)C=C5)CC4)(=O)=O)C=C3)=N2)N(CCC)C1=O
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Solubility
| Solvent | Max Conc. mg/mL | Max Conc. mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 54.3 | 100 |
Preparing Stock Solutions
for PSB 0788
The following data is based on the product molecular weight 543.04
Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.84 mL | 9.21 mL | 18.41 mL |
| 5 mM | 0.37 mL | 1.84 mL | 3.68 mL |
| 10 mM | 0.18 mL | 0.92 mL | 1.84 mL |
| 50 mM | 0.04 mL | 0.18 mL | 0.37 mL |
Calculators
Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Background References
References are publications that support the biological activity of the product.
Product Specific Notices for PSB 0788
For research use only
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