LY 2087101

Tocris Bioscience, part of Bio-Techne | Catalog # 4141

Allosteric potentiator of α7, α4β2 and α4β4 nAChRs
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Key Product Details

Description

Allosteric potentiator of α7, α4β2 and α4β4 nAChRs

View all Nicotinic (a7) Receptor Modulators »

Product Description

LY 2087101 is an allosteric potentiator of α7, α4β2 and α4β4 nAChRs; displays selectivity against α3β4 nAChRs. Thought to potentiate agonist-evoked α7 responses by binding within the nAChR transmembrane region.

Product Specifications

Molecular Weight

318.39

Formula

C15H11FN2OS2

Storage

Store at +4°C

Purity

≥98% (HPLC)

Chemical Name

[2-[(4-Fluorophenyl)amino]-4-methyl-5-thiazolyl]-3-thienylmethanone

CAS Number

913186-74-0

PubChem ID

11964458

InChI Key

PEAMDZVDNYENPN-UHFFFAOYSA-N

SMILES

O=C(C3=CSC=C3)C1=C(C)N=C(NC2=CC=C(F)C=C2)S1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 31.84 100
Ethanol 3.18 10

Preparing Stock Solutions for LY 2087101

The following data is based on the product molecular weight 318.39

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 3.14 mL 15.70 mL 31.41 mL
5 mM 0.63 mL 3.14 mL 6.28 mL
10 mM 0.31 mL 1.57 mL 3.14 mL
50 mM 0.06 mL 0.31 mL 0.63 mL

Calculators

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Background References

References are publications that support the biological activity of the product.

Product Documents for LY 2087101

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for LY 2087101

For research use only

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