L-798,106

Tocris Bioscience, part of Bio-Techne | Catalog # 3342

Potent and highly selective EP3 antagonist
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Key Product Details

Description

Potent and highly selective EP3 antagonist

View all Prostanoid Receptor Antagonists »

Product Description

L-798,106 is a potent and highly selective prostanoid EP3 receptor antagonist (Ki values are 0.3, 916, > 5000 and > 5000 nM at EP3, EP4, EP1 and EP2 respectively). Attenuates sulprostone-induced inhibition of EFS-evoked twitch and contractile responses in vivo.

Product Specifications

Molecular Weight

536.44

Formula

C27H22BrNO4S

Storage

Store at RT

Purity

≥98% (HPLC)

Chemical Name

N-[(5-Bromo-2-methoxyphenyl)sulfonyl]-3-[2-(2-naphthalenylmethyl)phenyl]-2-propenamide

CAS Number

244101-02-8

PubChem ID

15551229

InChI Key

ODTKFNUPVBULRJ-NTCAYCPXSA-N

SMILES

O=C(NS(C4=C(OC)C=CC(Br)=C4)(=O)=O)/C=C/C1=CC=CC=C1CC3=CC2=CC=CC=C2C=C3

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 53.64 100

Preparing Stock Solutions for L-798,106

The following data is based on the product molecular weight 536.44

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.86 mL 9.32 mL 18.64 mL
5 mM 0.37 mL 1.86 mL 3.73 mL
10 mM 0.19 mL 0.93 mL 1.86 mL
50 mM 0.04 mL 0.19 mL 0.37 mL

Calculators

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Background References

References are publications that support the biological activity of the product.

Product Documents for L-798,106

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for L-798,106

For research use only

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