GSK 0660

Tocris Bioscience, part of Bio-Techne | Catalog # 3433

Selective PPARδ antagonist
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Key Product Details

Description

Selective PPARδ antagonist

View all PPAR delta Receptor Inverse Agonists »

Product Description

GSK 0660 is a selective PPARδ antagonist (IC50 values are 0.155, > 10 and ≥ 10 μM at PPARδ, PPARα and PPARγ respectively). Exhibits inverse agonist effects when administered by itself.

Product Specifications

Molecular Weight

418.49

Formula

C19H18N2O5S2

Storage

Store at +4°C

Purity

≥98% (HPLC)

Chemical Name

3-[[[2-Methoxy-4-(phenylamino)phenyl]amino]sulfonyl]-2-thiophenecarboxylic acid methyl ester

CAS Number

1014691-61-2

PubChem ID

46233311

InChI Key

NDFKBGWLUHKMFY-UHFFFAOYSA-N

SMILES

O=S(NC1=C(OC)C=C(NC3=CC=CC=C3)C=C1)(C2=C(C(OC)=O)SC=C2)=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 41.85 100
Ethanol 4.18 10

Preparing Stock Solutions for GSK 0660

The following data is based on the product molecular weight 418.49

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.39 mL 11.95 mL 23.90 mL
5 mM 0.48 mL 2.39 mL 4.78 mL
10 mM 0.24 mL 1.19 mL 2.39 mL
50 mM 0.05 mL 0.24 mL 0.48 mL

Calculators

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Background References

References are publications that support the biological activity of the product.

Product Documents for GSK 0660

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for GSK 0660

For research use only

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