CGP 54626 hydrochloride
Tocris Bioscience a Bio-Techne Brand
Key Product Details
Description: | Potent and selective GABAB antagonist |
Chemical Name: | [S-(R*,R*)]-[3-[[1-(3,4-Dichlorophenyl)ethyl]amino]-2-hydroxypropyl](cyclohexylmethyl) phosphinic acid |
Purity: | ≥96% (HPLC) |
Molecular Weight: | 444.76 |
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Citations for CGP 54626 hydrochloride (33)
Citations are publications that use Bio-Techne products. Selected citations for CGP 54626 hydrochloride include:
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Martelli and Fiala
(2019)
Slow presynaptic mechanisms that mediate adaptation in the olfactory pathway of Drosophila.
Elife.
8
PMID: 31169499 -
Goutierre et al.
(2019)
KCC2 Regulates Neuronal Excitability and Hippocampal Activity via Interaction with Task-3 Channels.
Cell Rep.
28:91
PMID: 31269453 -
Lecat-Guillet
(2017)
FRET-based sensors unravel activation and allosteric modulation of the GABAB receptor.
Cell Chem Biol.
24(3):360
PMID: 28286129 -
Scholler
(2017)
HTS-compatible FRET-based conformational sensors clarify membrane receptor activation.
Nat Chem Biol.
13(4):372
PMID: 28135236 -
Zhang et al.
(2017)
Astrocytic Process Plasticity and IKKβ/NF-κB in Central Control of Blood Glucose, Blood Pressure, and Body Weight.
Cell Metab.
25:1091
PMID: 28467927 -
Xiao et al.
(2017)
Biased OXTergic Modulation of Midbrain DA Systems.
Neuron.
95:368
PMID: 28669546 -
Lin et al.
(2016)
Neuronal splicing regulator RBFOX3(NeuN) regulates adult hippocampal neurogenesis and synaptogenesis
PLoS One.
11:e0164164
PMID: 27701470 -
Zhang and Gaudry
(2016)
Functional integration of a serotonergic neuron in the Drosophila antennal lobe.
Elife.
5
PMID: 27572257 -
Bocchio et al.
(2015)
Increased serotonin transporter expression reduces fear and recruitment of parvalbumin interneurons of the amygdala.
Neuropsychopharmacology.
40:3015
PMID: 26052039 -
Zhang et al.
(2015)
GABAB receptor upregulates fragile X mental retardation protein expression in neurons.
Elife.
5:10468
PMID: 26020477 -
Chen et al.
(2015)
Morphine disinhibits glutamatergic input to VTA DA neurons and promotes DA neuron excitation.
J Neurosci.
4
PMID: 26208338 -
Kotecki et al.
(2015)
GIRK Channels Modulate Opioid-Induced Motor Activity in a Cell Type- and Subunit-Dependent Manner.
Proc Natl Acad Sci U S A.
35:7131
PMID: 25948263 -
Tachibana et al.
(2015)
Modification of Male Courtship Motivation by Olfactory Habituation via the GABAA Receptor in Drosophila melanogaster.
PLoS One.
10:e0135186
PMID: 26252206 -
Chumakov et al.
(2015)
Combining two repurposed drugs as a promising approach for Alzheimer's disease therapy.
Sci Rep.
5:7608
PMID: 25566747 -
Nagel et al.
(2015)
Synaptic and circuit mechanisms promoting broadband transmission of olfactory stimulus dynamics.
Nat Neurosci.
18:56
PMID: 25485755 -
Pfeffer et al.
(2013)
Inhibition of inhibition in visual cortex: the logic of connections between molecularly distinct interneurons.
Nat Neurosci.
16:1068
PMID: 23817549 -
Zhang et al.
(2013)
NE drives persistent activity in prefrontal cortex via synergistic α1 and α2 adrenoceptors.
PLoS One.
8:e66122
PMID: 23785477 -
Baloucoune et al.
(2012)
GABAB receptor subunit GB1 at the cell surface independently activates ERK1/2 through IGF-1R transactivation.
PLoS One.
7:e39698
PMID: 22761875 -
Werner et al.
(2011)
PKCγ is required for ethanol-induced increases in GABA(A) receptor α4 subunit expression in cultured cerebral cortical neurons.
J Biol Chem.
116:554
PMID: 21155805 -
Paz et al.
(2011)
A new mode of corticothalamic transmission revealed in the Gria4(-/-) model of absence epilepsy.
Proc Natl Acad Sci U S A.
14:1167
PMID: 21857658 -
Agarwal and Isacoff
(2011)
Specializations of a pheromonal glomerulus in the Drosophila olfactory system.
J Neurophysiol.
105:1711
PMID: 21289134 -
Tu et al.
(2010)
GABAB receptor activation protects neurons from apoptosis via IGF-1 receptor transactivation.
J Neurosci.
30:749
PMID: 20071540 -
Tani et al.
(2010)
Glutamine is required for persistent epileptiform activity in the disinhibited neocortical brain slice.
J Neurosci.
30:1288
PMID: 20107056 -
Ignell et al.
(2009)
Presynaptic peptidergic modulation of olfactory receptor neurons in Drosophila.
Br J Pharmacol.
106:13070
PMID: 19625621 -
Dacks et al.
(2009)
Serotonin modulates olfactory processing in the antennal lobe of Drosophila.
Nat Neurosci.
23:366
PMID: 19863268 -
Lörincz et al.
(2009)
ATP-dependent infra-slow (0.1 Hz) oscillations in thalamic networks.
PLoS One.
4:e4447
PMID: 19212445 -
Root et al.
(2008)
A presynaptic gain control mechanism fine-tunes olfactory behavior.
Neuron.
59:311
PMID: 18667158 -
Binet et al.
(2007)
Common structural requirements for heptahelical domain function in class A and class C G protein-coupled receptors.
J Neurogenet.
282:12154
PMID: 17310064 -
Shang et al.
(2007)
Excitatory local circuits and their implications for olfactory processing in the fly antennal lobe.
Cell.
128:601
PMID: 17289577 -
Gascon et al.
(2006)
GABA regulates dendritic growth by stabilizing lamellipodia in newly generated interneurons of the olfactory bulb.
J Neurosci.
26:12956
PMID: 17167085 -
Piet et al.
(2004)
Physiological contribution of the astrocytic environment of neurons to intersynaptic crosstalk.
Br J Pharmacol.
101:2151
PMID: 14766975 -
Dzitoyeva et al.
(2003)
Gamma-aminobutyric acid B receptor 1 mediates behavior-impairing actions of alcohol in Drosophila: adult RNA interference and pharmacological evidence.
Proc Natl Acad Sci U S A.
100:5485
PMID: 12692303 -
Wood et al.
(2000)
The human GABA(B1b) and GABA(B2) heterodimeric recombinant receptor shows low sensitivity to phaclofen and saclofen.
J Neurochem.
131:1050
PMID: 11082110
There are no citations that match your criteria.