CGP 42112

Tocris Bioscience, part of Bio-Techne | Catalog # 2569

Selective, high affinity AT2 ligand
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Key Product Details

Description

Selective, high affinity AT2 ligand

View all Angiotensin AT2 Receptor Ligands »

Product Description

CGP 42112 is a selective, high affinity angiotensin AT2 receptor ligand (Ki = 0.24 nM). Displays agonistic properties at proximal tubule AT2 receptors, causes Na+, K+-ATPase inhibition and sodium excretion. Antagonizes Ang-II induced contractions in rabbit aortic rings (IC50 = 1850 nM).

Product Specifications

Molecular Weight

1052.20

Formula

C52H69N13O11

Storage

Store at -20°C

Purity

≥95% (HPLC)

CAS Number

127060-75-7

PubChem ID

123794

InChI Key

UXGNARZDONUMMK-LRMQDCNJSA-N

SMILES

CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC1=CNC=N1)NC(=O)[C@H](CCCCNC(=O)[C@H](CCCNC(N)=N)NC(=O)OCC1=CC=CC=C1)NC(=O)[C@H](CC1=CC=C(O)C=C1)NC(=O)C1=CN=CC=C1)C(O)=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solubility Soluble to 1mg/ml in water

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Background References

References are publications that support the biological activity of the product.

Product Documents for CGP 42112

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for CGP 42112

For research use only

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