Key Product Details
Description: | β3 partial agonist. β1/β2 antagonist |
Chemical Name: | 4-[3-[(1,1-Dimethylethyl)amino]2-hydroxypropoxy]-1,3-dihydro-2H-benzimidazol-2-one hydrochloride |
Molecular Weight: | 315.8 |
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Citations for CGP 12177 hydrochloride (6)
Citations are publications that use Bio-Techne products. Selected citations for CGP 12177 hydrochloride include:
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Kilpatrick et al.
(2019)
Complex Formation between VEGFR2 and the β2-Adrenoceptor.
Cell Chem Biol.
2019;
PMID: 30956148 -
Gherbi et al.
(2015)
Negative cooperativity across β1-adrenoceptor homodimers provides insights into the nature of the secondary low-affinity CGP 12177 β1-adrenoceptor binding conformation.
FASEB J.
29:2859
PMID: 25837585 -
Stoddart et al.
(2015)
Application of BRET to monitor ligand binding to GPCRs.
Nat Methods.
12:661
PMID: 26030448 -
Littmann et al.
(2015)
Recruitment of β-arrestin 1 and 2 to the β2-adrenoceptor: analysis of 65 ligands.
Proc Natl Acad Sci U S A.
355:183
PMID: 26306764 -
Suárez et al.
(2014)
Oleoylethanolamide enhances β-adrenergic-mediated thermogenesis and white-to-brown adipocyte phenotype in epididymal white adipose tissue in rat.
Dis Model Mech.
7:129
PMID: 24159189 -
Gherbi et al.
(2014)
Detection of the secondary, low-affinity β1 -adrenoceptor site in living cells using the fluorescent CGP 12177 derivative BODIPY-TMR-CGP.
Br J Pharmacol.
171:5431
PMID: 25052258
There are no citations that match your criteria.