BD 1063 dihydrochloride

Citations are publications that use Bio-Techne products. Selected citations for BD 1063 dihydrochloride include:

• Cortés-Montero et al. (2019) The axonal motor neuropathy-related HINT1 protein is a zinc- and calmodulin-regulated cysteine SUMO protease. Antioxid Redox Signal. 2019;
  PMID: 31088288
• Sánchez-Blázquez et al. (2018) Sigma 1 Receptor Antagonists Inhibit Manic-Like Behaviors in Two Congenital Strains of Mice. Int J Neuropsychopharmacol. 21:938
  PMID: 29860313
• Rodríguez-Muñoz et al. (2018) Cannabidiol enhances MOR antinociception, diminishes NMDA-mediated seizures and reduces stroke damage via the sigma 1 receptor. Mol Brain. 11:51
  PMID: 30223868
• Sánchez-Blázquez et al. (2018) The Sigma-1 Receptor Antagonist, S1RA, Reduces Stroke Damage, Ameliorates Post-Stroke Neurological Deficits and Suppresses the Overexpression of MMP-9. Mol Neurobiol. 55:4940
  PMID: 28779350
• Rodríguez-Muñoz et al. (2015) The ON:OFF switch, σ1R-HINT1 protein, controls GPCR-NMDA receptor cross-regulation: implications in neurological disorders. Int J Neuropsychopharmacol. 6:35458
  PMID: 26461475
• Pabba et al. (2014) NMDA receptors are upregulated and trafficked to the plasma membrane after sigma-1 receptor activation in the rat hippocampus. J Neurosci. 34:11325
  PMID: 25143613
• Nguyen et al. (2014) Involvement of sigma-1 receptors in the antidepressant-like effects of dextromethorphan. PLoS One. 9:e89985
  PMID: 24587167
• Sánchez-Blázquez et al. (2014) The calcium-sensitive σ-1 receptor prevents cannabinoids from provoking glutamate NMDA receptor hypofunction: implications in antinociception and psychotic diseases. Nat Chem Biol. 17:1943
  PMID: 24485144
• Smith et al. (2014) A role for picomolar concentrations of pregnenolone sulfate in synaptic activity-dependent Ca²⁺ signaling and CREB activation. Mol Pharmacol. 86:390
  PMID: 25057049
• Pan et al. (2014) σ-1 receptor antagonism restores injury-induced decrease of voltage-gated Ca2+ current in sensory neurons. Oncotarget. 350:290
  PMID: 24891452
• Iñiguez et al. (2013) Inhibitory effects of sigma-2 receptor agonists on T lymphocyte activation. Front Pharmacol. 4:23
  PMID: 23494519
• Amer et al. (2013) Inhibition of endothelial cell Ca2+ entry and transient receptor potential channels by Sigma-1 receptor ligands. Br J Pharmacol. 168:1445
  PMID: 23121507
• Zhang et al. (2013) Methylphenidate enhances NMDA-receptor response in medial prefrontal cortex via sigma-1 receptor: a novel mechanism for methylphen. action. PLoS One. 7:e51910
  PMID: 23284812
• Kourrich et al. (2013) Dynamic interaction between sigma-1 receptor and Kv1.2 shapes neuronal and behavioral responses to cocaine. Cell. 152:236
  PMID: 23332758
• Fishback et al. (2012) A 96-well filtration method for radioligand binding analysis of σ receptor ligands. J Pharm Biomed Anal. 71:157
  PMID: 22910107
• Hiranita et al. (2011) Decreases in cocaine self-administration with dual inhibition of the DA transporter and σ receptors. J Pharmacol Exp Ther. 339:662
  PMID: 21859929
• Kurata et al. (2004) beta-OE, dehydroepiandrosterone, and dehydroepiandrosterone sulfate protect against N-MthD.-aspartate-induced neurotoxicity in rat hippocampal neurons by different mechanisms. J Pharmacol Exp Ther. 311:237
  PMID: 15175425

There are no citations that match your criteria.

Customer Images

• 
• (1)

• BD1063 binds to sigma-1 receptor

  Name: Timur Mavlyutov
  Species: Mouse
  Assay Type: In Vitro
  We used BD1063 compound as a sigma-1 receptor protector against photolabeling by radioactive iodoazidofenpropimorph in mouse spinal cord homogenate and saw good protective effect with concentration of 10uM.

• Use of BD 1063 in mouse brain slices

  Name: Jordan Yorgason
  Species: Mouse
  Assay Type: Ex Vivo
  Cell Line/Tissue: C57
  We used BD 1063 as a selective sigma antagonist to test if methamphetamine effects on dopamine release involved sigma receptor activation. BD 1063 (100nM) was applied before methamphetamine treatment. Drug was easy to use, and Tocris' recommendation on concentration for selectivity was useful for the study.
  PMID: 29185481 Reference
  

There are no reviews that match your criteria.