AM 251

Citations are publications that use Bio-Techne products. Selected citations for AM 251 include:

• Ellermann et al. (2020) Endocannabinoids inhibit the induction of virulence in enteric pathogens. Cell. 2020;
  PMID: 33031742
• Diniz et al. (2019) Dual mechanism of TRKB activation by anandamide through CB1 and TRPV1 receptors. PeerJ. 7:e6493
  PMID: 30809460
• Miranda et al. (2019) Cannabinoid Receptor 1 Blockade Attenuates Obesity and Adipose Tissue Type 1 Inflammation Through miR-30e-5p Regulation of Delta-Like-4 in Macrophages and Consequently Downregulation of Th1 Cells. Front Immunol. 10:1049
  PMID: 31134094
• Hu et al. (2019) Endocannabinoid Signaling Mediates Local Dendritic Coordination between Excitatory and Inhibitory Synapses. Cell Rep. 27:666
  PMID: 30995465
• Nasrallah et al. (2019) Routing Hippocampal Information Flow through Parvalbumin Interneuron Plasticity in Area CA2. Cell Rep. 27:86
  PMID: 30943417
• Alharris et al. (2019) Role of miRNA in the regulation of cannabidiol-mediated apoptosis in neuroblastoma cells. Oncotarget. 10:45
  PMID: 30713602
• Xiao et al. (2018) OXT functions as a spatiotemporal filter for excitatory synaptic inputs to VTA DA neurons. Elife. 7
  PMID: 29676731
• Johnston et al. (2018) Activity in nodose ganglia neurons after treatment with CP 55,940 and cholecystokinin. Physiol Rep. 6:e13927
  PMID: 30512249
• Song et al. (2018) Selective Role of RGS9-2 in Regulating Retrograde Synaptic Signaling of Indirect Pathway Medium Spiny Neurons in Dorsal Striatum. J Neurosci. 38:7120
  PMID: 30006367
• Eubler et al. (2018) Ca2+ Signaling and IL-8 Secretion in Human Testicular Peritubular Cells Involve the Cation Channel TRPV2. Int J Mol Sci. 19
  PMID: 30235802
• Han (2017) Cannabinoid receptor 1 contributes to sprouted innervation in endometrial ectopic growth through mitogen-activated protein kinase activation. Brain Res. 1663:132
  PMID: 28322749
• King-Himmelreich (2017) AMPK contributes to aerobic exercise-induced antinociception downstream of endocannabinoids. Neuropharmacology. 124:134
  PMID: 28479394
• Saliba (2017) AM404, paracetamol metabolite, prevents prostaglandin synthesis in activated microglia by inhibiting COX activity. J Neuroinflammation. 14(1):246
  PMID: 29237478
• Zhang (2017) Orphan nuclear receptor ERRγ is a key regulator of human fibrinogen gene expression. PLoS One. 12(7):e0182141
  PMID: 28750085
• Fatahi (2017) Involvement of cannabinoid system in the nucleus accumbens on delay-based decision making in the rat. Behav Brain Res.. 337:107
  PMID: 28987618
• Leroy et al. (2017) Input-Timing-Dependent Plasticity in the Hippocampal CA2 Region and Its Potential Role in Social Memory. Neuron. 95:1089
  PMID: 28823730
• Shang et al. (2016) Δ 9-Tetrahydrocannabinol Reverses TNFα-induced Increase in Airway Epithelial Cell Permeability through CB 2 Receptors Biochemical Pharmacology. 2016;
  PMID: 27641813
• Krohn et al. (2016) Abnormal cannabidiol attenuates experimental colitis in mice, promotes wound healing and inhibits neutrophil recruitment. J Inflamm (Lond). 13:21
  PMID: 27418880
• Cui et al. (2016) Endocannabinoid dynamics gate spike-timing dependent depression and potentiation. Elife. 5:e13185
  PMID: 26920222
• Blaha et al. (2016) Impaired Excitatory Neurotransmission in the Urinary Bladder from the Obese Zucker Rat: Role of Cannabinoid Receptors. PLoS One. 11:e0157424
  PMID: 27285468
• Xie et al. (2016) Up-regulation of immunomodulatory effects of mouse bone-marrow derived mesenchymal stem cells by tetrahydrocannabinol pre-treatment involving cannabinoid receptor CB2. Oncotarget. 7:6436
  PMID: 26824325
• Yu et al. (2016) Dentate cannabinoid-sensitive interneurons undergo unique and selective strengthening of mutual synaptic inhibition in experimental epilepsy. Neurobiol Dis. 89:23
  PMID: 26804027
• Malek et al. (2015) Anandamide, Acting via CB2 Receptors, Alleviates LPS-Induced Neuroinflammation in Rat Primary Microglial Cultures. Neural Plast. 2015:130639
  PMID: 26090232
• Zhang et al. (2015) Anoctamin Calcium-Activated Chloride Channels May Modulate Inhibitory Transmission in the Cerebellar Cortex. PLoS One. 10:e0142160
  PMID: 26558388
• Yang et al. (2015) Cannabinoid receptor CB2 is involved in tetrahydrocannabinol-induced anti-inflammation against lipopolysaccharide in MG-63 cells. Sci Rep. 2015:362126
  PMID: 25653478
• Liu et al. (2015) Involvement of GluR2 up-regulation in neuroprotection by electroacupuncture pretreatment via cannabinoid CB1 receptor in mice. Nutr Diabetes. 5:9490
  PMID: 25830356
• Vähätalo et al. (2015) Role of the endocannabinoid system in obesity induced by neuropeptide Y overexpression in noradrenergic neurons. Mol Cell Neurosci. 5:e151
  PMID: 25915740
• Zhou et al. (2015) Regional effects of endocannabinoid, BDNF and FGF receptor signalling on neuroblast motility and guidance along the rostral migratory stream. Nat Commun. 64:32
  PMID: 25481343
• Dincheva et al. (2015) FAAH genetic variation enhances fronto-amygdala function in mouse and human. Nat Commun. 6:6395
  PMID: 25731744
• Lenkey et al. (2015) Tonic endocannabinoid-mediated modulation of GABA release is independent of the CB1 content of axon terminals. Sci Rep. 6:6557
  PMID: 25891347
• Smith et al. (2015) The Effects of the Endocannabinoids Anandamide and 2-Arachidonoylglycerol on Human Osteoblast Proliferation and Differentiation. Proc Natl Acad Sci U S A. 10:e0136546
  PMID: 26414859
• Bowles et al. (2015) A peripheral endocannabinoid mechanism contributes to glucocorticoid-mediated metabolic syndrome. Mol Pharmacol. 112:285
  PMID: 25535367
• Stanley et al. (2015) Cannabidiol causes endothelium-dependent vasorelaxation of human mesenteric arteries via CB1 activation. Front Cell Neurosci. 107:568
  PMID: 26092099
• Martin et al. (2015) Endocannabinoids Mediate Muscarinic Acetylcholine Receptor-Dependent Long-Term Depression in the Adult Medial Prefrontal Cortex. Br J Pharmacol. 9:457
  PMID: 26648844
• Krishnan and Chatterjee (2015) Differential immune mechanism to HIV-1 Tat variants and its regulation by AEA [corrected]. PLoS One. 5:9887
  PMID: 25943894
• Parvathy and Masocha (2015) Coadministration of indomet. and MinCyc attenuates established PacT.-induced neuropathic thermal hyperalgesia: Involvement of cannabinoid CB1 receptors. J Neurosci. 5:10541
  PMID: 26085115
• Wang et al. (2015) Activation of cannabinoid receptor 1 inhibits increased bladder activity induced by nerve growth factor. Neurosci Lett. 589:19
  PMID: 25575795
• Arrabal et al. (2015) Pharmacological Blockade of Cannabinoid CB1 Receptors in Diet-Induced Obesity Regulates Mitochondrial Dihydrolipoamide Dehydrogenase in Muscle. PLoS One. 10:e0145244
  PMID: 26671069
• Bashashati et al. (2015) Inhibiting endocannabinoid biosynthesis: a novel approach to the treatment of constipation. Br J Pharmacol. 172:3099
  PMID: 25684407
• Ma et al. (2015) Mitochondrial CB1 receptor is involved in ACEA-induced protective effects on neurons and mitochondrial functions. Sci Rep. 5:12440
  PMID: 26215450
• Stornaiuolo et al. (2015) Endogenous vs Exogenous Allosteric Modulators in GPCRs: A dispute for shuttling CB1 among different membrane microenvironments. Sci Rep. 5:15453
  PMID: 26482099
• Szabó et al. (2014) Presynaptic calcium channel inhibition underlies CB1 cannabinoid receptor-mediated suppression of GABA release. Mediators Inflamm. 34:7958
  PMID: 24899717
• Alpár et al. (2014) Endocannabinoids modulate cortical development by configuring Slit2/Robo1 signalling. J Neurosci. 5:4421
  PMID: 25030704
• Tortoriello et al. (2014) Miswiring the brain: △9-tetrahydrocannabinol disrupts cortical development by inducing an SCG10/stathmin-2 degradation pathway. Proc Natl Acad Sci U S A. 33:668
  PMID: 24469251
• Hassanzadeh and Rostami (2014) CB1 cannabinoid receptors are involved in neuroleptic-induced enhancement of brain neurotensin. J Neurosci. 17:181
  PMID: 24847420
• Costa et al. (2014) 2-arachidonoylglycerol effects in cytotrophoblasts: metabolic enzymes expression and apoptosis in BeWo cells. Reproduction. 147:301
  PMID: 24324206
• Cass et al. (2014) CB1 cannabinoid receptor stimulation during adolescence impairs the maturation of GABA function in the adult rat prefrontal cortex. Mol Psychiatry. 19:536
  PMID: 24589887
• Xu et al. (2014) Hippocampal metaplasticity is required for the formation of temporal associative memories. J Neurosci. 34:16762
  PMID: 25505329
• Kury et al. (2014) Effects of the endogenous cannabinoid anandamide on voltage-dependent sodium and calcium channels in rat ventricular myocytes. Br J Pharmacol. 171:3485
  PMID: 24758718
• Sreevalsan and Safe (2013) The cannabinoid WIN 55,212-2 decreases specificity protein transcription factors and the oncogenic cap protein eIF4E in colon cancer cells. Mol Cancer Ther. 12:2483
  PMID: 24030632
• Malenczyk et al. (2013) CB1 cannabinoid receptors couple to focal adhesion kinase to control Ins release. J Biol Chem. 288:32685
  PMID: 24089517
• Abush and Akirav (2013) Cannabinoids ameliorate impairments induced by chronic stress to synaptic plasticity and short-term memory. Neuropsychopharmacology. 38:1521
  PMID: 23426383
• Cao et al. (2013) Cannabinoid HU210 protects isolated rat stomach against impairment caused by serum of rats with experimental acute pancreatitis. PLoS One. 7:e52921
  PMID: 23285225
• Wargent et al. (2013) The cannabinoid δ(9)-tetrahydrocannabivarin (THCV) ameliorates Ins sensitivity in two mouse models of obesity. Nutr Diabetes. 3:e68
  PMID: 23712280
• Chanda et al. (2013) Hepatic cannabinoid receptor type 1 mediates alcohol-induced regulation of bile acid enzyme genes expression via CREBH. PLoS One. 8:e68845
  PMID: 23894352
• Benz et al. (2013) Expression and functional relevance of cannabinoid receptor 1 in Hodgkin lymphoma. PLoS One. 8:e81675
  PMID: 24349109
• Keimpema et al. (2013) Diacylglycerol lipase α manipulation reveals developmental roles for intercellular endocannabinoid signaling. Nat Commun. 3:2093
  PMID: 23806960
• Baca et al. (2013) Gene-environment interactions affect long-term depression (LTD) through changes in DA receptor affinity in Snap25 deficient mice. Brain Res. 1532:85
  PMID: 23939223
• Hayase (2013) Working memory- and anxiety-related behavioral effects of repeated nicotine as a stressor: the role of cannabinoid receptors. BMC Neurosci. 14:20
  PMID: 23394117
• Li et al. (2013) Inhibition of fatty acid amide hydrolase activates Nrf2 signalling and induces heme oxygenase 1 transcription in breast cancer cells. Br J Pharmacol. 170:489
  PMID: 23347118
• Duncan et al. (2013) Cannabinoid 1 receptors are critical for the innate immune response to TLR4 stimulation. Am J Physiol Regul Integr Comp Physiol. 305:R224
  PMID: 23739343
• Rossi et al. (2013) The cannabinoid receptor type 2 as mediator of mesenchymal stromal cell immunosuppressive properties. PLoS One. 8:e80022
  PMID: 24312195
• Ganon-Elazar and Akirav (2012) Cannabinoids prevent the development of behavioral and endocrine alterations in a rat model of intense stress. Neuropsychopharmacology. 37:456
  PMID: 21918506
• Guida et al. (2012) Salvinorin A reduces mechanical allodynia and spinal neuronal hyperexcitability induced by peripheral formalin injection. Mol Pain. 8:60
  PMID: 22913292
• Tozzi et al. (2012) A2A adenosine receptor antagonism enhances synaptic and motor effects of cocaine via CB1 cannabinoid receptor activation. PLoS One. 7:e38312
  PMID: 22715379
• Caiati et al. (2012) Developmental regulation of CB1-mediated spike-time dependent depression at immature mossy fiber-CA3 synapses. Sci Rep. 2:285
  PMID: 22368777
• Stern et al. (2012) On disruption of fear memory by reconsolidation blockade: evidence from cannabidiol treatment. Neuropsychopharmacology. 37:2132
  PMID: 22549120
• Tumati et al. (2012) Repeated mor. treatment-mediated hyperalgesia, allodynia and spinal glial activation are blocked by co-administration of a selective cannabinoid receptor type-2 agonist. J Neuroimmunol. 244:23
  PMID: 22285397
• Laricchiuta et al. (2012) CB1 receptor autoradiographic characterization of the individual differences in approach and avoidance motivation. PLoS One. 7:e42111
  PMID: 22848724
• Brents et al. (2012) Monohydroxylated metabolites of the K2 synthetic cannabinoid JWH-073 retain intermediate to high cannabinoid 1 receptor (CB1R) affinity and exhibit neutral antagonist to partial agonist activity. Biochem Pharmacol. 83:952
  PMID: 22266354
• Liu et al. (2012) Betulinic acid targets YY1 and ErbB2 through cannabinoid receptor-dependent disruption of microRNA-27a:ZBTB10 in breast cancer. Mol Cancer Ther. 11:1421
  PMID: 22553354
• Casarotto et al. (2012) Opposing roles for cannabinoid receptor type-1 (CB1) and transient receptor potential vanilloid type-1 channel (TRPV1) on the modulation of panic-like responses in rats. Pain. 37:478
  PMID: 21937980
• Niu et al. (2012) Effects of gonadal hormones on the peripheral cannabinoid receptor 1 (CB1R) system under a myositis condition in rats. J Pharmacol Exp Ther. 153:2283
  PMID: 22940464
• Chanda et al. (2012) Activation of cannabinoid receptor type 1 (Cb1r) disrupts hepatic Ins receptor signaling via cyclic AMP-response element-binding protein H (Crebh)-mediated induction of Lipin1 gene. Br J Pharmacol. 287:38041
  PMID: 22989885
• Gonzalez-Islas et al. (2012) Tonic and transient endocannabinoid regulation of AMPAergic miniature postsynaptic currents and homeostatic plasticity in embryonic motor networks. Sci Rep. 32:13597
  PMID: 23015449
• Giordano et al. (2012) TRPV1-dependent and -independent alterations in the limbic cortex of neuropathic mice: impact on glial caspases and pain perception. Cereb Cortex. 22:2495
  PMID: 22139792
• Laricchiuta et al. (2012) Differences in spontaneously avoiding or approaching mice reflect differences in CB1-mediated signaling of dorsal striatal transmission. PLoS One. 7:e33260
  PMID: 22413007
• Merighi et al. (2012) Cannabinoid CB(2) receptors modulate ERK-1/2 kinase signalling and NO release in microglial cells stimulated with bacterial lipopolysaccharide. Br J Pharmacol. 165:1773
  PMID: 21951063
• Peterfi et al. (2012) Endocannabinoid-mediated long-term depression of afferent excitatory synapses in hippocampal pyramidal cells and GABAergic interneurons. J Neurosci. 32:14448
  PMID: 23055515
• Sideris et al. (2012) A Role for the Cannabinoid 1 Receptor in Neuronal Differentiation of Adult Spinal Cord Progenitors in vitro is Revealed through Pharmacological Inhibition and Genetic Deletion. Front Neurosci. 6:4
  PMID: 22291615
• Tauber et al. (2012) Regulation of MMP-9 by a WIN-binding site in the monocyte-macrophage system independent from cannabinoid receptors. PLoS One. 7:e48272
  PMID: 23139770
• Hamtiaux et al. (2012) The association of N-palmitoylethanolamine with the FAAH inhibitor URB597 impairs melanoma growth through a supra-additive action. BMC Cancer. 12:92
  PMID: 22429826
• Aydin et al. (2012) Nicotine-induced anxiety-like behavior in a rat model of the novelty-seeking phenotype is associated with long-lasting neuropeptidergic and neuroplastic adaptations in the amygdala: effects of the cannabinoid receptor 1 antagonist AM251. Neuropharmacology. 63:1335
  PMID: 22959963
• Baur et al. (2012) The cannabinoid CB1 receptor antagonists rim. (SR141716) and AM251 directly potentiate GABA(A) receptors. Br J Pharmacol. 165:2479
  PMID: 21470203
• Merighi et al. (2012) Cannabinoid CB(2) receptor attenuates morphine-induced inflammatory responses in activated microglial cells. Br J Pharmacol. 166:2371
  PMID: 22428664
• Méndez-D?az et al. (2012) The endocannabinoid system modulates the valence of the emotion associated to food ingestion. Addict Biol. 17:725
  PMID: 21182571
• Li and Burrell (2011) Associative, bidirectional changes in neural signaling utilizing NMDA receptor- and endocannabinoid-dependent mechanisms. Learn Mem. 18:545
  PMID: 21844187
• Brents et al. (2011) Phase I hydroxylated metabolites of the K2 synthetic cannabinoid JWH-018 retain in vitro and in vivo cannabinoid 1 receptor affinity and activity. PLoS One. 6:e21917
  PMID: 21755008
• Crespillo et al. (2011) Expression of the cannabinoid system in muscle: effects of a high-fat diet and CB1 receptor blockade. Biochem J. 433:175
  PMID: 20955176
• Pan et al. (2011) Alterations of endocannabinoid signaling, synaptic plasticity, learning, and memory in monoacylglycerol lipase knock-out mice. J Cell Biol. 31:13420
  PMID: 21940435
• Hassanzadeh and Hassanzadeh (2011) The Role of the Endocannabinoids in Suppression of the Hypothalamic-pituitary-adrenal Axis Activity by dox. J Leukoc Biol. 14:414
  PMID: 23493814
• Negrete et al. (2011) The antinociceptive effects of JWH-015 in chronic inflammatory pain are produced by nitric oxide-cGMP-PKG-KATP pathway activation mediated by opioids. PLoS One. 6:e26688
  PMID: 22031841
• Guidali et al. (2011) Cannabinoid CB1 receptor antagonism prevents neurochemical and behavioural deficits induced by chronic phencyclidine. Int J Neuropsychopharmacol. 14:17
  PMID: 20196921
• Segev and Akirav (2011) Differential effects of cannabinoid receptor agonist on social discrimination and contextual fear in amygdala and hippocampus. Learn Mem. 18:254
  PMID: 21447623
• Samineni et al. (2011) Post-ictal analgesia in genetically epilepsy-prone rats is induced by audiogenic seizures and involves cannabinoid receptors in the periaqueductal gray. Brain Res. 1389:177
  PMID: 21439272
• Thompson and Perkel (2011) Endocannabinoids mediate synaptic plasticity at glutamatergic synapses on spiny neurons within a basal ganglia nucleus necessary for song learning. J Neurophysiol. 105:1159
  PMID: 21177997
• Sousa et al. (2011) Regulation of hippocampal cannabinoid CB1 receptor actions by adenosine A1 receptors and chronic caffeine administration: implications for the effects of δ9-tetrahydrocannabinol on spatial memory. Neuropsychopharmacology. 36:472
  PMID: 20927050
• Ruby et al. (2011) Acute overactive endocannabinoid signaling induces glucose intolerance, hepatic steatosis, and novel cannabinoid receptor 1 responsive genes. PLoS One. 6:e26415
  PMID: 22073164
• Novellis et al. (2011) The blockade of the transient receptor potential vanilloid type 1 and fatty acid amide hydrolase decreases symptoms and central sequelae in the medial prefrontal cortex of neuropathic rats. Mol Pain. 7:7
  PMID: 21241462
• Hamtiaux et al. (2011) Increasing antiproliferative properties of endocannabinoids in N1E-115 neuroblastoma cells through inhibition of their metabolism. PLoS One. 6:e26823
  PMID: 22046372
• Yuan and Burrell (2010) Endocannabinoid-dependent LTD in a nociceptive synapse requires activation of a presynaptic TRPV-like receptor. J Neurophysiol. 104:2766
  PMID: 20884761
• Jiang et al. (2010) The maturation of GABAergic transmission in visual cortex requires endocannabinoid-mediated LTD of inhibitory inputs during a critical period. Neuron. 66:248
  PMID: 20435001
• Buznikov et al. (2010) A putative 'pre-nervous' endocannabinoid system in early echinoderm development. Dev Neurosci. 32:1
  PMID: 19907129
• Mair et al. (2010) Interaction between anandamide and sphingosine-1-phosphate in mediating vasorelaxation in rat coronary artery. Br J Pharmacol. 161:176
  PMID: 20718749
• Atkinson et al. (2010) Regulation of the hypothalamic-pituitary-adrenal axis circadian rhythm by endocannabinoids is sexually diergic. Endocrinology. 151:3720
  PMID: 20534730
• Schlosburg et al. (2010) Chronic monoacylglycerol lipase blockade causes functional antagonism of the endocannabinoid system. Nat Neurosci. 13:1113
  PMID: 20729846
• Henstridge et al. (2010) GPR55 ligands promote receptor coupling to multiple signalling pathways. Br J Pharmacol. 160:604
  PMID: 20136841
• Curto-Reyes et al. (2010) Spinal and peripheral analgesic effects of the CB2 cannabinoid receptor agonist AM1241 in two models of bone cancer-induced pain. Br J Pharmacol. 160:561
  PMID: 20233215
• Acuna-Goycolea et al. (2010) Cannabinoids excite circadian clock neurons. J Neurosci. 30:10061
  PMID: 20668190
• Farkas et al. (2010) Retrograde endocannabinoid signaling reduces GABAergic synaptic transmission to gonadotropin-releasing hormone neurons. J Biol Chem. 151:5818
  PMID: 20926585
• Jones et al. (2010) Cannabidiol displays antiepileptiform and antiseizure properties in vitro and in vivo. Cereb Cortex. 332:569
  PMID: 19906779
• Ho et al. (2010) Endocannabinoid modulation of hyperaemia evoked by physiologically relevant stimuli in the rat primary somatosensory cortex. Neuropsychopharmacology. 160:736
  PMID: 20590576
• Hao et al. (2010) The cannabinoid WIN55,212-2 protects against oxidized LDL-induced inflammatory response in murine macrophages. Iran J Basic Med Sci. 51:2181
  PMID: 20305287
• Bhaskaran and Smith (2010) Effects of TRPV1 activation on synaptic excitation in the dentate gyrus of a mouse model of temporal lobe epilepsy. Endocrinology. 223:529
  PMID: 20144892
• Wamsteeker et al. (2010) Repeated stress impairs endocannabinoid signaling in the paraventricular nucleus of the hypothalamus. J Neurosci. 30:11188
  PMID: 20720126
• Huang et al. (2010) A refractory period for rejuvenating GABAergic synaptic transmission and ocular dominance plasticity with dark exposure. J Neurosci. 30:16636
  PMID: 21148002
• Losonczy et al. (2010) Network mechanisms of theta related neuronal activity in hippocampal CA1 pyramidal neurons. Nat Neurosci. 13:967
  PMID: 20639875
• Touriño et al. (2010) THC Prevents MDMA Neurotoxicity in Mice. PLoS One. 5:e9143
  PMID: 20174577
• Hoffman et al. (2010) Control of cannabinoid CB1 receptor function on glutamate axon terminals by endogenous adenosine acting at A1 receptors. J Neurosci. 30:545
  PMID: 20071517
• Godlewski et al. (2010) Inhibitor of fatty acid amide hydrolase normalizes cardiovascular function in hypertension without adverse metabolic effects. Chem Biol. 17:1256
  PMID: 21095576
• Zhang et al. (2010) Cannabinoid CB1 receptor facilitation of substance P release in the rat spinal cord, measured as neurokinin 1 receptor internalization. Eur J Neurosci. 31:225
  PMID: 20074214
• Garzón et al. (2009) Gz mediates the long-lasting desensitization of brain CB1 receptors and is essential for cross-tolerance with mor. Mol Pain. 5:11
  PMID: 19284549
• Mendiguren and Pineda (2009) Effect of the CB(1) receptor antagonists rim. and AM251 on the firing rate of dorsal raphe nucleus neurons in rat brain slices. Br J Pharmacol. 158:1579
  PMID: 19845674
• Tjen-A-Looi et al. (2009) Processing cardiovascular information in the vlPAG during electroacupuncture in rats: roles of endocannabinoids and GABA. J Appl Physiol (1985). 106:1793
  PMID: 19325030
• Fraga et al. (2009) Endogenous cannabinoids induce fever through the activation of CB1 receptors. Neuropsychopharmacology. 157:1494
  PMID: 19681872
• Meuth et al. (2009) The neuroprotective impact of the leak potassium channel TASK1 on stroke development in mice. Exp Neurol. 33:42675
  PMID: 18930826
• Wallace et al. (2009) PKCε regulates behavioral sensitivity, binding and tolerance to the CB1 receptor agonist WIN55,212-2. Iran J Basic Med Sci. 34:1733
  PMID: 19158669
• Ho and Gardiner (2009) Acute hypertension reveals depressor and vasodilator effects of cannabinoids in conscious rats. Br J Pharmacol. 156:94
  PMID: 19133994
• Pan et al. (2009) Blockade of 2-arachidonoylglycerol hydrolysis by selective monoacylglycerol lipase inhibitor 4-nitrophenyl 4-(dibenzo[d][1,3]dioxol-5-yl(hydroxy)methyl)piperidine-1-carboxylate (JZL184) Enhances retrograde endocannabinoid signaling. J Pharmacol Exp Ther. 331:591
  PMID: 19666749
• Pacheco et al. (2009) Central antinociception induced by mu-opioid receptor agonist morphine, but not delta- or kappa-, is mediated by cannabinoid CB1 receptor. Br J Pharmacol. 158:225
  PMID: 19594755
• Shen et al. (2008) Dichotomous DArgic control of striatal synaptic plasticity. Science. 321:848
  PMID: 18687967
• Gibson et al. (2008) TRPV1 channels mediate long-term depression at synapses on hippocampal interneurons. Neuron. 57:746
  PMID: 18341994
• Melis et al. (2008) Endogenous fatty acid ethanolamides suppress nicotine-induced activation of mesolimbic DA neurons through nuclear receptors. J Neurosci. 28:13985
  PMID: 19091987
• Potenzieri et al. (2008) The cannabinoid receptor agonist, WIN 55, 212-2, attenuates tumor-evoked hyperalgesia through peripheral mechanisms. Brain Res. 1215:69
  PMID: 18486111
• Börner et al. (2008) Analysis of promoter regions regulating basal and interleukin-4-inducible expression of the human CB1 receptor gene in T lymphocytes. Eur J Pharmacol. 73:1013
  PMID: 18156315
• Georgieva et al. (2008) Unique agonist-bound cannabinoid CB1 receptor conformations indicate agonist specificity in signaling. Br J Pharmacol. 581:19
  PMID: 18162180
• Giannini et al. (2008) Activation of cannabinoid receptors prevents antigen-induced asthma-like reaction in guinea pigs. Br J Pharmacol. 12:2381
  PMID: 18266975
• Desroches et al. (2008) Modulation of the anti-nociceptive effects of 2-arachidonoyl glycerol by peripherally administered FAAH and MGL inhibitors in a neuropathic pain model. Eur J Neurosci. 155:913
  PMID: 18695638
• Naguib et al. (2008) MDA7: a novel selective agonist for CB2 receptors that prevents allodynia in rat neuropathic pain models. Br J Pharmacol. 155:1104
  PMID: 18846037
• Xia et al. (2008) Electroacupuncture of 2?hz has a rewarding effect: evidence from a conditioned place preference study in rats. Evid Based Complement Alternat Med. 2011:730514
  PMID: 18955347
• Ruby et al. (2008) Overactive endocannabinoid signaling impairs apolipoprotein E-mediated clearance of triglyceride-rich lipoproteins. Proc Natl Acad Sci U S A. 105:14561
  PMID: 18794527
• Wilson et al. (2008) Repeated cannabinoid injections into the rat periaqueductal gray enhance subsequent mor. antinociception. Neuropharmacology. 55:1219
  PMID: 18723035
• Durakoglugil and Orer (2008) Cannabinoid receptor activation in the nucleus tractus solitaries produces baroreflex-like responses in the rat. Int J Biomed Sci. 4:229
  PMID: 23675095
• Toscano et al. (2008) Altered GABAergic neurotransmission is associated with increased kainate-induced seizure in prostaglandin-endoperoxide synthase-2 deficient mice. Brain Res Bull. 75:598
  PMID: 18355636
• Huang et al. (2008) Roles of endocannabinoids in heterosynaptic long-term depression of excitatory synaptic transmission in visual cortex of young mice. J Neurosci. 28:7074
  PMID: 18614676
• Pacheco et al. (2008) The mu-opioid receptor agonist morphine, but not agonists at delta- or kappa-opioid receptors, induces peripheral antinociception mediated by cannabinoid receptors. Br J Pharmacol. 154:1143
  PMID: 18469844
• Kim et al. (2008) Interactions between CB(1) receptors and TRPV1 channels mediated by 12-HPETE are cytotoxic to mesencephalic DArgic neurons. Br J Pharmacol. 155:253
  PMID: 18552868
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• CB1R antagonist AM251 (5 µM)

  Name: Kang Peng
  Species: Mouse
  Assay Type: In Vitro
  Cell Line/Tissue: auditory brainstem（MNTB）
  bath application of the CB1R antagonist AM251 (5 µM)

There are no reviews that match your criteria.