MDR1/ABCB1 Products
6 results for "MDR1/ABCB1" in Products
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MDR1/ABCB1 Products
6 results for "MDR1/ABCB1" in Products
Selective MRP1 and P-gp inhibitor
Chemical Name : | N-[3-(4-Morpholinyl)propyl]-5,7-diphenylpyrazolo[1,5-a]pyrimidine-3-carboxamide |
Purity : | ≥95% (HPLC) |
P-gp and BCRP inhibitor
Alternate Names : | GF 120918 |
Chemical Name : | N-[4-[2-(3,4-Dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)ethyl]phenyl]-9,10-dihydro-5-methoxy-9-oxo-4-acridinecarboxamide hydrochloride |
Purity : | ≥98% (HPLC) |
Potent P-glycoprotein (P-gp) inhibitor
Chemical Name : | N-[2-[[[4-[2-(3,4-dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)ethyl]phenyl]amino]carbonyl]-4,5-dimethoxyphenyl]-3-quinolinecarbxamide dihydrochloride |
Purity : | ≥98% (HPLC) |
High affinity P-gp inhibitor
Alternate Names : | LY 335979 |
Chemical Name : | (αR)-4-[(1aα,6α,10bα)-1,1-Difluoro-1,1a,6,10b-tetrahydrodibenzo[a,e]cyclopropa[c]cyclohepten-6-yl]-α-[(5-quinolinyloxy)methyl]-1-piperazineethanol trihydrochloride |
Purity : | ≥97% (HPLC) |