Dopamine D3 Receptor Agonists: Small Molecules and Peptides
DRD3 is the D3 subtype of the five (D1-D5) dopamine receptors. The activity of the D3 subtype receptor is mediated by G proteins which inhibit adenylyl cyclase. It is localized to the limbic areas of the brain, which are associated with cognitive, emotional, and endocrine functions. Genetic variations may be associated with susceptibility to hereditary essential tremor 1. Alternative splicing results in transcript variants encoding different isoforms. This variant represents the predominant transcript and encodes the longer isoform (a).
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Dopamine D3 Receptor Agonists: Small Molecules and Peptides
DRD3 is the D3 subtype of the five (D1-D5) dopamine receptors. The activity of the D3 subtype receptor is mediated by G proteins which inhibit adenylyl cyclase. It is localized to the limbic areas of the brain, which are associated with cognitive, emotional, and endocrine functions. Genetic variations may be associated with susceptibility to hereditary essential tremor 1. Alternative splicing results in transcript variants encoding different isoforms. This variant represents the predominant transcript and encodes the longer isoform (a).
4 results for "Dopamine D3 Receptor Agonists Small Molecules and Peptides" in Products
Selective D3 agonist
Chemical Name : | (S)-2-Amino-4,5,6,7-tetrahydro-6-(propylamino)benzothiazole dihydrochloride |
Purity : | ≥99% (HPLC) |
Dopamine D3 receptor biased agonist
Chemical Name : | 2-chloro-α-methyl-benzenepropanamine hydrochloride |
Purity : | ≥98% (HPLC) |
High affinity D3 agonist (D3 ≥ D2 > D4)
Chemical Name : | (4aR,10bR)-3,4a,4,10b-Tetrahydro-4-propyl-2H,5H-[1]benzopyrano-[4,3-b]-1,4-oxazin-9-ol hydrochloride |
Purity : | ≥98% (HPLC) |
D2 and D3 agonist
Alternate Names : | N 0923 |
Chemical Name : | (6S)-5,6,7,8-Tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-1-naphthalenol hydrochloride |
Purity : | ≥99% (HPLC) |