Ocinaplon

Name: Ocinaplon
Brand: Tocris Bioscience
SKU: 4410

Tocris Bioscience, part of Bio-Techne | Catalog # 4410

COA / SDS

GABAA modulator; anxiolytic

Discontinued Product

4410 has been discontinued. View all GABA-A Receptor Modulators products.

Key Product Details

Description:	GABA_A modulator; anxiolytic
Chemical Name:	2-Pyridinyl[7-(4-pyridinyl)pyrazolo[1,5-a]pyrimidin-3-yl]methanone
Purity:	≥98% (HPLC)
Molecular Weight:	301.3

View Full Technical Details for Ocinaplon

Technical Data
Citations

Biological Activity for Ocinaplon

Ocinaplon is a modulator of GABA_A receptors. Displays modest selectivity for GABA_A α₁ receptors; displays partial agonist activity at α2-, α3- and α5-containing receptors. Exhibits anxiolytic activity.

Technical Data for Ocinaplon

M. Wt	301.3
Formula	C₁₇H₁₁N₅O
Storage	Store at +4°C
Purity	≥98% (HPLC)
CAS Number	96604-21-6
PubChem ID	216456
InChi Key	OQJFBUOFGHPMSR-UHFFFAOYSA-N
Smiles	O=C(C4=CC=CC=N4)C2=C1N=CC=C(C3=CC=NC=C3)N1N=C2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

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References for Ocinaplon

References are publications that support the biological activity of the product.

Lippa Selective anxiolysis produced by ocinaplon, a GABA_A receptor modulator. Proc.Natl.Acad.Sci.USA 2005 PMID: 15870187
Rupprecht GABA_A receptors as targets for novel anxiolytic drugs. World J.Biol.Psychiatry 2006 PMID: 17071543
Mirza Comparative cue generalization profiles of L-838,417, SL651498, zolpidem, CL218,872, ocinaplon, bretazenil, ZopiC., and various benzodiazepines in chlordiazep. and zol. drug discrimination. J.Pharmacol.Exp.Ther. 2006 PMID: 16339395

Ocinaplon

Tocris Bioscience, part of Bio-Techne | Catalog # 4410

Key Product Details

Biological Activity for Ocinaplon

Technical Data for Ocinaplon

Molarity Calculator

Dilution Calculator

Reconstitution Calculator

References for Ocinaplon

Product Documents for Ocinaplon

COA

Certificate of Analysis

SDS

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