N-Benzylnaltrindole hydrochloride

Name: N -Benzylnaltrindole hydrochloride
Brand: tocris
SKU: 0754

Catalog # 0754

Datasheet / COA / SDS

Order Information

Bio-Techne Corporation

tel: (612) 379-2956

tel: (800) 343-7475 (free phone)

customercare.na@bio-techne.com

Shipping Information

$35 to United States

Products in stock will be shipped in 1-3 business days unless specified.

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Key Product Details

Description:	Selective non-peptide δ₂ antagonist
Chemical Name:	1'-Benzyl-17-(cyclopropylmethyl)-6,7-didehydro-4,5a-epoxy-3,14-dihydroxyindolo[2',3':6,7]morphinan hydrochloride

View Full Technical Details for N-Benzylnaltrindole hydrochloride

Technical Data
Citations / Reviews

Biological Activity

Potent δ₂-selective opioid receptor antagonist with a long duration of action in vivo.

Technical Data

M. Wt	541.09
Formula	C₃₃H₃₂N₂O₃.HCl
Storage	Store at RT
CAS Number	1206487-81-1
PubChem ID	90479740
InChi Key	KDEBSUYWJUBPCB-ZHYTUUPESA-N
Smiles	O[C@@]24[C@]3([C@@H]8C(N6CC7=CC=CC=C7)=C(C5=C6C=CC=C5)C4)C1=C(O8)C(O)=CC=C1CC2N(CC9CC9)CC3.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Solubility

	Solvent	Max Conc. mg/mL	Max Conc. mM
Solubility
Solubility	DMSO	54.11	100

Preparing Stock Solutions

The following data is based on the product molecular weight 541.09.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.85 mL	9.24 mL	18.48 mL
5 mM	0.37 mL	1.85 mL	3.70 mL
10 mM	0.18 mL	0.92 mL	1.85 mL
50 mM	0.04 mL	0.18 mL	0.37 mL

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Reconstitution Calculator

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References

References are publications that support the biological activity of the product.

Korlipara N-Benzylnaltrindoles as long acting δ-opioid receptor antagonists. J.Med.Chem. 1994 PMID: 8021928