Deltorphin I
Tocris Bioscience, part of Bio-Techne | Catalog # 4591
Potent δ agonist
Discontinued Product
4591 has been discontinued.
View all delta Opioid Receptor Agonists products.
Product Description
Deltorphin I is a potent δ-opioid receptor agonist (IC50 = 0.5 nM in human granulocytes). Exhibits a high rate of blood-brain barrier penetrance.Product Specifications
Molecular Weight
768.87
Formula
C37H52N8O10
Storage
Store at -20°C
CAS Number
122752-15-2
PubChem ID
10055958
InChI Key
CJAORFIPPWIGPG-QXYJMILXSA-N
SMILES
[H]N[C@@H](CC1=CC=C(O)C=C1)C(=O)N[C@H](C)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](C(C)C)C(=O)NCC(N)=O
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Solubility
| Solubility | Soluble to 1mg/ml in 20% formic acid |
Calculators
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Background References
References are publications that support the biological activity of the product.
- Erspamer Deltorphins: a family of naturally occurring peptides with high affinity and selectivity for δ opioid binding sites. Proc.Natl.Acad.Sci.USA 1989 PMID: 2544892
- Fiori Deltorphin transport across the blood-brain barrier. Proc.Natl.Acad.Sci.USA 1997 PMID: 9256506
- Stefano [D-Ala2]Deltorphin I binding and pharmacological evidence for a special subtype of δ opioid receptor on human and invertebrate immune cells. Proc.Natl.Acad.Sci.USA 1992 PMID: 1329092
Product Specific Notices for Deltorphin I
For research use only
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