BMS 470539 dihydrochloride

Tocris Bioscience, part of Bio-Techne | Catalog # 4053

Potent, selective MC1 receptor agonist
Discontinued Product
4053 has been discontinued. View all Melanocortin Receptor Agonists products.

Key Product Details

Description

Potent, selective MC1 receptor agonist

View all Melanocortin Receptor Agonists »

Product Description

BMS 470539 dihydrochloride is a potent, selective melanocortin MC1 receptor agonist (IC50 = 120 nM). Exhibits anti-inflammatory properties following ischemia-reperfusion in the vasculature. Inhibits leukocyte trafficking.

Product Specifications

Molecular Weight

632.62

Formula

C32H41N5O4.2HCl

Storage

Desiccate at RT

Purity

≥98% (HPLC)

Chemical Name

1-[1-(3-Methyl-L-histidyl-O-methyl-D-tyrosyl)-4-phenyl-4-piperidinyl]-1-butanone dihydrochloride

CAS Number

2341796-82-3

PubChem ID

60210130

InChI Key

DUAOBJHRUKFKIH-YDVFRNEYSA-N

SMILES

O=C(N2CCC(C(CCC)=O)(C4=CC=CC=C4)CC2)[C@H](NC([C@@H](N)CC3=CN=CN3C)=O)CC1=CC=C(OC)C=C1.Cl.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 63.26 100
DMSO 63.26 100

Preparing Stock Solutions for BMS 470539 dihydrochloride

The following data is based on the product molecular weight 632.62

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.58 mL 7.90 mL 15.81 mL
5 mM 0.32 mL 1.58 mL 3.16 mL
10 mM 0.16 mL 0.79 mL 1.58 mL
50 mM 0.03 mL 0.16 mL 0.32 mL

Calculators

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Product Documents for BMS 470539 dihydrochloride

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for BMS 470539 dihydrochloride

For research use only

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